SCHEMBL4786471

SCHEMBL4786471

CCOC(=O)[C@H](Cc1ccc(Nc2ncccc2NC(=O)C(F)(F)F)cc1)NC1=CC(=O)C12CCCCC2

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 14/20 0.44
ITGA4 P13612 14/20 0.44
CYP3A4 P08684 3/20 0.35
CYP2C9 P11712 3/20 0.35
ELANE P08246 1/20 0.33
BRD4 O60885 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4739188 0.93 ITGB1 (0.45) ITGB1ITGA4CYP3A4CYP2C9ELANE
SCHEMBL4737693 0.86 ITGB1 (0.43) ITGB1ITGA4CYP3A4CYP2C9ELANE
SCHEMBL4735581 0.85 ITGB1 (0.46) ITGB1ITGA4CYP3A4CYP2C9ELANE
SCHEMBL4733927 0.84 ITGB1 (0.43) ITGB1ITGA4CYP3A4CYP2C9
SCHEMBL4733784 0.83 MAPT (0.52) ITGB1ITGA4
SCHEMBL3832796 0.79 ITGB1 (0.47) ITGB1ITGA4CYP3A4CYP2C9ELANE
SCHEMBL4737637 0.78 ITGB1 (0.42) ITGB1ITGA4ELANE
SCHEMBL4736687 0.77 MAPT (0.48) ITGB1ITGA4
SCHEMBL4735983 0.76 ITGA4 (0.47) ITGB1ITGA4CYP3A4CYP2C9ELANE
SCHEMBL4750224 0.76 ITGB1 (0.44) ITGB1ITGA4CYP3A4ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008064830-A1 BICYCLIC AND HETEROBICYCLIC DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR PHARMACEUTICAL USES UCB PHARMA, S.A. (BE) 2008-06-05 WO claimed
WO-2008064830-A1 BICYCLIC AND HETEROBICYCLIC DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR PHARMACEUTICAL USES UCB PHARMA, S.A. (BE) 2008-06-05 WO disclosed