SCHEMBL4786704

SCHEMBL4786704

Cc1cc2ccn(C(=O)O)c(=O)c2c(-c2ccc(F)cc2)n1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AKR1B10 O60218 4/20 0.40
PARP1 P09874 1/20 0.37
NTRK1 P04629 1/20 0.36
NTRK2 Q16620 1/20 0.36
ALDH1A1 P00352 2/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
TP53 P04637 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36
DHODH Q02127 2/20 0.36
CES2 O00748 1/20 0.36
ADORA2A P29274 2/20 0.36
ADORA2B P29275 1/20 0.36
ADORA1 P30542 1/20 0.36
KDM4C Q9H3R0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4788032 0.87 NTRK1 (0.39) AKR1B10PARP1NTRK1NTRK2ALDH1A1
SCHEMBL4747721 0.82 KDM4C (0.41) ALDH1A1NPC1RAB9ATP53KDM4E
SCHEMBL4787999 0.80 MAPT (0.39) AKR1B10PARP1ALDH1A1KDM4EMAPT
SCHEMBL5815996 0.79 ALDH1A1 (0.37) ALDH1A1NPC1RAB9ATP53KDM4E
SCHEMBL4751131 0.78 KDM4C (0.38) ALDH1A1NPC1RAB9ATP53KDM4E
SCHEMBL27778077 0.76 ALDH1A1 (0.40) AKR1B10ALDH1A1HSD17B10DHODH
SCHEMBL4788527 0.75 MAPK14 (0.42) TP53MAPT
SCHEMBL4747281 0.71 EGFR (0.46) ALDH1A1TP53MAPTHSD17B10
SCHEMBL27778063 0.70 MAPK14 (0.40) KDM4EHSD17B10KDM4C
SCHEMBL4750216 0.69 GRIA1 (0.40) NTRK2ALDH1A1NPC1RAB9ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008123755-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTAM TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO claimed
WO-2008123755-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTAM TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO disclosed