SCHEMBL4787624

SCHEMBL4787624

Cc1nc(-c2ccccc2)n(C)c1C(=O)N=C(N)N

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.49
SLC9A1 P19634 9/20 0.48
PLAU P00749 3/20 0.48
SLC9A2 Q9UBY0 1/20 0.43
ASIC3 Q9UHC3 1/20 0.41
SLC9A5 Q14940 1/20 0.40
DHODH Q02127 1/20 0.40
PTGER1 P34995 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4784404 0.88 SLC9A1 (0.51) SLC9A1SLC9A5
SCHEMBL4786226 0.84 SLC9A1 (0.52) SLC9A1
SCHEMBL2682845 0.83 CYP1A2 (0.55) CYP1A2DHODHPTGER1
SCHEMBL4788479 0.81 SLC9A1 (0.49) SLC9A1
SCHEMBL11312831 0.80 CYP1A2 (0.58) CYP1A2DHODHPTGER1
SCHEMBL4787618 0.75 CYP1A2 (0.47) CYP1A2DHODHPTGER1
Hydrochloric Acid SCHEMBL6312712 0.74 PLAU (0.47) SLC9A1PLAUSLC9A2ASIC3
SCHEMBL4787413 0.73 TP53 (0.51) SLC9A1SLC9A5
SCHEMBL4786806 0.71 ALDH1A1 (0.48) SLC9A1
Hydrochloric Acid SCHEMBL6313857 0.70 PLAU (0.52) SLC9A1PLAUSLC9A2ASIC3SLC9A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008111794-A1 4-METHYLIMIDAZOL-5-YLCARBONYLGUANIDINE DERIVATIVES, PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF, PREPARATION METHOD, AND PHARMACEUTICAL COMPOSITIONS FOR THE PREVENTION AND TREATMENT OF THE ISCHEMIC HEART DISEASES CONTAINING THE SAME AS AN ACTIVE INGREDIENT KOREA RESERACH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2008-09-18 WO disclosed