SCHEMBL4787983

SCHEMBL4787983

CC(C)c1cc(NC(=O)Nc2ccc(Oc3ccnc(N)c3)cc2F)n(-c2ccc(Cl)cc2)n1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 9/20 0.61
MAPK13 O15264 2/20 0.51
BRAF P15056 11/20 0.49
KCNJ6 P48051 1/20 0.47
KCNJ5 P48544 1/20 0.47
KCNJ3 P48549 1/20 0.47
PLK4 O00444 1/20 0.47
ACOX3 O15254 1/20 0.47
MAP3K7 O43318 1/20 0.47
DYRK3 O43781 1/20 0.47
JAK2 O60674 1/20 0.47
ERN1 O75460 1/20 0.47
RPS6KA4 O75676 1/20 0.47
STK10 O94804 1/20 0.47
MAP4K4 O95819 1/20 0.47
ABL1 P00519 1/20 0.47
RAF1 P04049 1/20 0.47
NTRK1 P04629 1/20 0.47
LCK P06239 1/20 0.47
FYN P06241 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4686310 0.93 MAPK14 (0.65) MAPK14MAPK13BRAFPLK4ACOX3
SCHEMBL4648264 0.89 MAPK14 (0.59) MAPK14MAPK13BRAFPLK4ACOX3
SCHEMBL4647702 0.87 MAPK14 (0.79) MAPK14MAPK13BRAFKCNJ6KCNJ5
SCHEMBL4648677 0.86 MAPK14 (0.57) MAPK14MAPK13BRAFKCNJ6KCNJ5
SCHEMBL2025093 0.86 MAPK14 (0.65) MAPK14MAPK13BRAFPLK4ACOX3
SCHEMBL2246332 0.85 ABL1 (0.51) MAPK14MAPK13BRAFKCNJ6KCNJ5
SCHEMBL4648705 0.83 BRAF (0.55) MAPK14MAPK13BRAFKCNJ6KCNJ5
SCHEMBL4745379 0.83 MAPK14 (0.66) MAPK14MAPK13BRAFKCNJ6KCNJ5
SCHEMBL4746824 0.83 MAPK14 (0.77) MAPK14MAPK13BRAFPLK4ACOX3
SCHEMBL4647243 0.82 MAPK14 (0.79) MAPK14MAPK13BRAFPLK4ACOX3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960394-A2 PYRAZOLYL UREA DERIVATIVES USEFUL IN THE TREATMENT OF CANCER Bayer HealthCare AG (DE) 2008-08-27 EP disclosed
WO-2007059202-A2 PYRAZOLYL UREA DERIVATIVES USEFUL IN THE TREATMENT OF CANCER BAYER HEALTHCARE AG (DE) 2007-05-24 WO disclosed