SCHEMBL4788935

SCHEMBL4788935

CNc1c(C(=O)Nc2cc(NC(=O)c3cc(-n4cnc(C)c4)cc(C(F)(F)F)c3)ccc2C)cnc2[nH]ccc12

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 2/20 0.63
MAPT P10636 1/20 0.61
KDM4E B2RXH2 1/20 0.59
POLB P06746 1/20 0.59
RECQL P46063 1/20 0.59
MAPK14 Q16539 1/20 0.54
MAP3K20 Q9NYL2 1/20 0.54
MAP3K7 O43318 1/20 0.54
MAP4K2 Q12851 1/20 0.54
RAF1 P04049 4/20 0.52
EPHB2 P29323 1/20 0.52
BRAF P15056 4/20 0.52
ABL1 P00519 3/20 0.52
HCK P08631 2/20 0.52
BCR P11274 2/20 0.52
LYN P07948 2/20 0.52
EGFR P00533 1/20 0.52
LCK P06239 1/20 0.52
FYN P06241 1/20 0.52
YES1 P07947 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4788930 0.91 MAPK14 (0.53) CSF1RMAPTKDM4EPOLBRECQL
SCHEMBL4787141 0.88 CSF1R (0.67) CSF1RMAPTKDM4EPOLBRECQL
SCHEMBL14026838 0.86 BRAF (0.66) CSF1RMAPK14MAP3K7MAP4K2RAF1
SCHEMBL4789921 0.86 KDR (0.48) CSF1RMAPK14RAF1BRAFABL1
SCHEMBL4788638 0.85 CSF1R (0.69) CSF1RMAPTKDM4EPOLBRECQL
SCHEMBL4788677 0.84 CSF1R (0.56) CSF1RMAPK14MAP3K20MAP3K7MAP4K2
SCHEMBL4788891 0.84 CSF1R (0.61) CSF1RMAPK14RAF1BRAFABL1
SCHEMBL13708168 0.84 CSF1R (0.61) CSF1RMAPTKDM4EPOLBRECQL
SCHEMBL14069752 0.82 MAPT (0.59) CSF1RMAPTKDM4EPOLBRECQL
SCHEMBL19376837 0.81 CSF1R (0.74) CSF1RMAPTKDM4EPOLBRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008144253-A1 PROTEIN KINASE INHIBITORS AND METHODS FOR USING THEREOF IRM LLC (BM) 2008-11-27 WO disclosed
WO-2008144253-A1 PROTEIN KINASE INHIBITORS AND METHODS FOR USING THEREOF IRM LLC (BM) 2008-11-27 WO disclosed