SCHEMBL4789010

SCHEMBL4789010

C[N+]1(CCc2ccc3c(c2)OCO3)CC2C(CCC(C#N)(c3ccccc3)c3ccccc3)C2C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
TSHR P16473 1/20 0.35
ACHE P22303 1/20 0.35
TAAR1 Q96RJ0 1/20 0.34
HTR2A P28223 2/20 0.34
HTR2C P28335 2/20 0.34
HTR2B P41595 2/20 0.34
TRPM8 Q7Z2W7 1/20 0.34
CALM1 P0DP23 1/20 0.34
CYP3A4 P08684 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
DRD2 P14416 2/20 0.33
DRD4 P21917 2/20 0.33
OPRM1 P35372 2/20 0.33
DRD3 P35462 2/20 0.33
CHRM3 P20309 2/20 0.33
CCR1 P32246 2/20 0.33
CYP2D6 P10635 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4790311 0.94 CCR1 (0.36) ALDH1A1TSHRACHETAAR1HTR2A
SCHEMBL4788471 0.91 CHRM3 (0.37) ALDH1A1TSHRTAAR1HTR2AHTR2C
SCHEMBL4788452 0.87 TSHR (0.36) ALDH1A1TSHRACHETAAR1HTR2A
SCHEMBL4790212 0.85 MAPT (0.36) ALDH1A1TSHRTAAR1TRPM8CALM1
SCHEMBL4789864 0.85 CHRM3 (0.37) ALDH1A1TSHRACHETRPM8TDP1
SCHEMBL4788570 0.84 CHRM3 (0.38) ALDH1A1TSHRACHETAAR1CHRM3
SCHEMBL4788351 0.82 ALDH1A1 (0.34) ALDH1A1TSHRACHETAAR1HTR2A
SCHEMBL4790547 0.81 ALDH1A1 (0.42) ALDH1A1TSHRKCNA3
SCHEMBL4789873 0.80 CHRM3 (0.39) ALDH1A1TSHRACHETAAR1HTR2A
SCHEMBL4789383 0.80 CHRM3 (0.36) ALDH1A1TSHRTAAR1HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008117229-A1 MUSCARINIC RECEPTOR ANTAGONISTS RANBAXY LABORATORIES LIMITED (IN) 2008-10-02 WO claimed
WO-2008117229-A1 MUSCARINIC RECEPTOR ANTAGONISTS RANBAXY LABORATORIES LIMITED (IN) 2008-10-02 WO disclosed