SCHEMBL4789249

SCHEMBL4789249

CN1CCN(c2cccc3c2C[C@H](NC(=O)c2ccc(C(F)(F)F)nc2)CC3)CC1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.56
SCN9A Q15858 5/20 0.56
SCN5A Q14524 4/20 0.56
HTR1A P08908 1/20 0.44
HTR1D P28221 1/20 0.44
HTR1B P28222 1/20 0.44
MTNR1A P48039 1/20 0.44
MTNR1B P49286 1/20 0.44
FAAH O00519 1/20 0.43
ACKR3 P25106 2/20 0.41
KMT2A Q03164 1/20 0.39
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39
TRPV1 Q8NER1 1/20 0.39
HPGDS O60760 2/20 0.38
SLC6A5 Q9Y345 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4887320 0.87 SCN9A (0.74) KCNH2SCN9ASCN5AMTNR1AMTNR1B
SCHEMBL7025761 0.87 KCNH2 (0.55) KCNH2SCN9ASCN5AMTNR1AMTNR1B
SCHEMBL6820338 0.87 KCNH2 (0.55) KCNH2SCN9ASCN5AMTNR1AMTNR1B
SCHEMBL6820334 0.87 KCNH2 (0.55) KCNH2SCN9ASCN5AMTNR1AMTNR1B
SCHEMBL4788895 0.85 KCNH2 (0.49) KCNH2SCN9ASCN5AMTNR1AMTNR1B
SCHEMBL7030282 0.84 MEN1 (0.55) KCNH2SCN9ASCN5AMTNR1AMTNR1B
SCHEMBL7031232 0.84 MEN1 (0.55) KCNH2SCN9ASCN5AMTNR1AMTNR1B
SCHEMBL4788755 0.84 SCN9A (0.75) KCNH2SCN9ASCN5AHPGDS
SCHEMBL7029805 0.84 KCNH2 (0.54) KCNH2SCN9ASCN5AMTNR1AMTNR1B
SCHEMBL7019156 0.84 KCNH2 (0.54) KCNH2SCN9ASCN5AMTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008130323-A1 NOVEL 8-PIPERAZINE-TETRAHYDRONAPHTALENE DERIVATIVES FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2008-10-30 WO disclosed