SCHEMBL4789293

SCHEMBL4789293

N#Cc1cccc2c1CCN(C(=O)C1CCCCC1C(=O)NC1(C#N)CC1)C2

nearest known ligand 0.68

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSK P43235 18/20 0.68
CTSB P07858 3/20 0.58
CTSS P25774 2/20 0.58
KCNH2 Q12809 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8106184 1.00 CTSK (0.68) CTSKCTSBCTSSKCNH2
SCHEMBL4787930 0.90 CTSK (0.69) CTSKCTSBCTSSKCNH2
SCHEMBL8100198 0.90 CTSK (0.69) CTSKCTSBCTSSKCNH2
SCHEMBL8108549 0.88 CTSK (0.70) CTSKCTSBCTSSKCNH2
SCHEMBL4789866 0.87 CTSK (0.70) CTSKCTSBCTSSKCNH2
SCHEMBL8111663 0.83 CTSK (0.69) CTSKCTSBCTSSKCNH2
SCHEMBL4757161 0.83 CTSK (0.69) CTSKCTSBCTSSKCNH2
SCHEMBL8108547 0.82 CTSK (0.67) CTSKCTSBCTSSKCNH2
SCHEMBL8091663 0.81 CTSK (1.00) CTSKCTSB
SCHEMBL2248479 0.81 CTSK (1.00) CTSKCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001128-A1 1,2-CYCL0HEXANE DICARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed