SCHEMBL4789900

SCHEMBL4789900

CC(C)(C)N(CCc1cc(Br)n(S(=O)(=O)c2cccnc2)c1)C(=O)O.COc1ccc(F)c(-c2cc(CC(NC(=O)O)C(C)(C)C)cn2S(=O)(=O)c2cccnc2)c1

nearest known ligand 0.32

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MMP9 P14780 6/20 0.32
MMP1 P03956 4/20 0.32
MMP13 P45452 4/20 0.32
NAMPT P43490 1/20 0.31
ADAM17 P78536 3/20 0.31
HTR6 P50406 4/20 0.30
CHRNB4 P30926 1/20 0.30
CHRNA3 P32297 1/20 0.30
KEAP1 Q14145 1/20 0.30
NFE2L2 Q16236 1/20 0.30
LMNA P02545 1/20 0.30
MMP2 P08253 1/20 0.30
USP30 Q70CQ3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4789904 0.93 MMP1 (0.36) MMP9MMP1MMP13NAMPTADAM17
SCHEMBL4792892 0.90
SCHEMBL4791519 0.89 NAMPT (0.32) NAMPT
SCHEMBL1278276 0.89 NAMPT (0.38) MMP9MMP1MMP13NAMPTHTR6
SCHEMBL4422713 0.87
SCHEMBL4791384 0.86
Fumaric Acid SCHEMBL4791584 0.82 NAMPT (0.35) MMP9MMP1MMP13NAMPTHTR6
SCHEMBL4792897 0.82 PTGDR2 (0.33) NAMPTADAM17CHRNB4CHRNA3
SCHEMBL4791521 0.81 NAMPT (0.36) MMP9MMP1MMP13NAMPT
SCHEMBL4791781 0.81 PDE10A (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919865-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2008-05-14 EP disclosed
WO-2007026916-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-03-08 WO disclosed