SCHEMBL4789904

SCHEMBL4789904

CC(C)(C)C(Cc1cc(Br)n(S(=O)(=O)c2cccnc2)c1)NC(=O)O.COc1ccc(F)c(-c2cc(CC(NC(=O)O)C(C)(C)C)cn2S(=O)(=O)c2cccnc2)c1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 3/20 0.36
MMP9 P14780 3/20 0.36
MMP13 P45452 3/20 0.36
NAMPT P43490 2/20 0.35
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
LMNA P02545 1/20 0.34
HTR6 P50406 8/20 0.34
DRD2 P14416 3/20 0.33
HTR2A P28223 2/20 0.33
ADAM17 P78536 2/20 0.33
GRM2 Q14416 1/20 0.33
CTSA P10619 1/20 0.33
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
MEN1 O00255 1/20 0.33
POLB P06746 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1278276 0.96 NAMPT (0.38) MMP1MMP9MMP13NAMPTCHRNB4
SCHEMBL4789900 0.93 MMP9 (0.32) MMP1MMP9MMP13NAMPTCHRNB4
Fumaric Acid SCHEMBL4791584 0.89 NAMPT (0.35) MMP1MMP9MMP13NAMPTCHRNB4
SCHEMBL4792897 0.88 PTGDR2 (0.33) NAMPTCHRNB4CHRNA3ADAM17POLB
SCHEMBL4791521 0.87 NAMPT (0.36) MMP1MMP9MMP13NAMPT
SCHEMBL1157389 0.87 PTGDR2 (0.37) NAMPTCHRNB4CHRNA3POLB
SCHEMBL1156754 0.86 HSD17B10 (0.38) MMP1MMP9MMP13ADAM17
SCHEMBL4422719 0.85 PTGDR2 (0.33) ADAM17
Carbamic Acid SCHEMBL4791644 0.84 HSD17B10 (0.36) MMP1MMP9MMP13ADAM17
SCHEMBL1278508 0.83 FPR1 (0.34) NAMPTCHRNB4CHRNA3POLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919865-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2008-05-14 EP disclosed
WO-2007026916-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-03-08 WO disclosed