SCHEMBL4792897

SCHEMBL4792897

CC(C)(C)C(Cc1cc(-c2ccncc2F)n(S(=O)(=O)c2cccnc2)c1)NC(=O)O.CC(C)(C)C(Cc1cc(Br)n(S(=O)(=O)c2cccnc2)c1)NC(=O)O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 1/20 0.33
FPR1 P21462 1/20 0.32
HSD17B10 Q99714 1/20 0.32
CHRNB2 P17787 1/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31
CHRNA4 P43681 1/20 0.31
TSHR P16473 2/20 0.31
ALDH1A1 P00352 2/20 0.31
POLB P06746 1/20 0.31
ABCC9 O60706 1/20 0.30
ABCC8 Q09428 1/20 0.30
KCNJ11 Q14654 1/20 0.30
KCNJ8 Q15842 1/20 0.30
ADAM17 P78536 1/20 0.30
HTT P42858 2/20 0.30
GAA P10253 1/20 0.30
GFER P55789 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
NAMPT P43490 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1278508 0.95 FPR1 (0.34) PTGDR2FPR1HSD17B10CHRNB2CHRNB4
SCHEMBL4792892 0.92
SCHEMBL1156754 0.89 HSD17B10 (0.38) FPR1HSD17B10CHRNB2CHRNA4TSHR
SCHEMBL4422719 0.89 PTGDR2 (0.33) PTGDR2FPR1HSD17B10ADAM17
SCHEMBL4789904 0.88 MMP1 (0.36) CHRNB4CHRNA3POLBADAM17SMN1; SMN2
Carbamic Acid SCHEMBL4791644 0.88 HSD17B10 (0.36) FPR1HSD17B10TSHRALDH1A1ABCC9
Fumaric Acid SCHEMBL4791575 0.88 FPR1 (0.31) FPR1HSD17B10POLB
Fumaric Acid SCHEMBL4791570 0.88 FPR1 (0.31) FPR1HSD17B10POLB
SCHEMBL1156935 0.87 POLB (0.39) PTGDR2FPR1HSD17B10CHRNB2CHRNB4
SCHEMBL4791390 0.87 HSD17B10 (0.31) PTGDR2HSD17B10ADAM17

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919865-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2008-05-14 EP disclosed
WO-2007026916-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-03-08 WO disclosed