SCHEMBL4790214

SCHEMBL4790214

C=CCN(C(=O)OCc1ccccc1)c1cc(C)cc(C(=O)O)c1NS(=O)(=O)CCC

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 1/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
GAA P10253 2/20 0.36
MAPT P10636 2/20 0.36
MEN1 O00255 1/20 0.36
HPGD P15428 1/20 0.36
KMT2A Q03164 1/20 0.36
HSD17B10 Q99714 1/20 0.36
ACLY P53396 2/20 0.34
F13A1 P00488 1/20 0.34
TGM2 P21980 1/20 0.34
TGM1 P22735 1/20 0.34
CCR5 P51681 2/20 0.33
MCL1 Q07820 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4651960 0.73 ALDH1A1 (0.49) ALDH1A1MAPTHPGDKMT2ALMNA
SCHEMBL2526014 0.72 ALDH1A1 (0.36) KDM4EALDH1A1GAAMAPTHPGD
SCHEMBL4790217 0.72 ALDH1A1 (0.34) ALDH1A1MAPTHPGDF13A1TGM2
SCHEMBL2529528 0.71 ALDH1A1 (0.38) ALDH1A1MAPTMEN1HPGDKMT2A
SCHEMBL4874190 0.69 SMN1; SMN2 (0.38) ALDH1A1MAPTHPGDMCL1LMNA
SCHEMBL3081849 0.67 HCAR2 (0.47) ALDH1A1MAPTMEN1HPGDKMT2A
SCHEMBL2527725 0.67 MAPT (0.40) KDM4EALDH1A1GAAMAPTHPGD
SCHEMBL15375412 0.67 HCAR2 (0.42) ALDH1A1MAPTHPGDKMT2ATGM2
SCHEMBL2531116 0.64 KMT2A (0.38) KDM4EALDH1A1GAAMAPTMEN1
SCHEMBL2526958 0.64 ALDH1A1 (0.41) ALDH1A1MAPTMEN1HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968954-A1 MACROCYCLIC COMPOUNDS USEFUL AS BACE INHIBITORS Novartis AG (CH) 2008-09-17 EP disclosed
WO-2007077004-A1 MACROCYCLIC COMPOUNDS USEFUL AS BACE INHIBITORS NOVARTIS AG (CH) 2007-07-12 WO disclosed