SCHEMBL4790217

SCHEMBL4790217

C=CCN(C(=O)OCc1ccccc1)c1c(N)c(C(=O)O)cc(C)c1S(=O)(=O)CCC

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.34
LMNA P02545 1/20 0.33
MAPK1 P28482 2/20 0.33
CYP3A4 P08684 1/20 0.33
TSHR P16473 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
F13A1 P00488 1/20 0.32
TGM2 P21980 1/20 0.32
TGM1 P22735 1/20 0.32
CCR5 P51681 3/20 0.32
MAPT P10636 2/20 0.32
HPGD P15428 1/20 0.31
F2 P00734 1/20 0.31
ELANE P08246 1/20 0.31
CTSG P08311 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4874190 0.72 SMN1; SMN2 (0.38) ALDH1A1LMNAMAPK1TSHRTDP1
SCHEMBL4790214 0.72 METAP2 (0.36) ALDH1A1LMNAF13A1TGM2TGM1
SCHEMBL2529528 0.69 ALDH1A1 (0.38) ALDH1A1TSHRF13A1TGM2TGM1
SCHEMBL4651960 0.69 ALDH1A1 (0.49) ALDH1A1LMNAMAPK1CYP3A4TSHR
SCHEMBL3081849 0.67 HCAR2 (0.47) ALDH1A1LMNAMAPK1TSHRTDP1
SCHEMBL4699372 0.65 MAPT (0.36) ALDH1A1LMNACYP3A4TSHRTDP1
SCHEMBL2527725 0.65 MAPT (0.40) ALDH1A1LMNAMAPK1CYP3A4TSHR
SCHEMBL2531116 0.64 KMT2A (0.38) ALDH1A1LMNATSHRTDP1L3MBTL1
SCHEMBL4756433 0.64 KDM4E (0.42) ALDH1A1MAPK1CYP3A4TSHRTDP1
SCHEMBL2526958 0.64 ALDH1A1 (0.41) ALDH1A1TSHRTDP1L3MBTL1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968954-A1 MACROCYCLIC COMPOUNDS USEFUL AS BACE INHIBITORS Novartis AG (CH) 2008-09-17 EP disclosed
WO-2007077004-A1 MACROCYCLIC COMPOUNDS USEFUL AS BACE INHIBITORS NOVARTIS AG (CH) 2007-07-12 WO disclosed