SCHEMBL4790340

SCHEMBL4790340

C[C](c1cc(-c2cscc2C)n(S(=O)(=O)c2cccnc2)c1)C(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.42
CYP2E1 P05181 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2B6 P20813 1/20 0.42
CYP2C19 P33261 1/20 0.42
CHRM5 P08912 1/20 0.33
NAPRT Q6XQN6 1/20 0.33
POLB P06746 1/20 0.32
KMT2A Q03164 1/20 0.32
CSNK2A2 P19784 1/20 0.32
CSNK2B P67870 1/20 0.32
KDM4E B2RXH2 1/20 0.32
USP2 O75604 1/20 0.31
HTT P42858 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
LMNA P02545 2/20 0.31
MAPT P10636 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4793151 0.88 PTGES2 (0.35) CHRM5NAPRTPOLBKMT2AKDM4E
Methylamine SCHEMBL28371746 0.82 CYP2A6 (0.45) CYP2A6CYP2E1CYP3A4CYP2D6CYP2C9
SCHEMBL4792177 0.82 CYP2A6 (0.37) CYP2A6CHRM5NAPRTPOLBKMT2A
SCHEMBL4791372 0.80 GBA1 (0.40) CYP2A6CYP2E1CYP3A4CYP2C9CYP2B6
SCHEMBL4790343 0.80 CYP2E1 (0.39) CYP2A6CYP2E1CYP3A4CYP2D6CYP2C9
SCHEMBL4793065 0.79 PTGS2 (0.44)
SCHEMBL14828747 0.78 CYP2E1 (0.41) CYP2A6CYP2E1CYP3A4CYP2D6CYP2C9
SCHEMBL193717 0.77 CYP2E1 (0.40) CYP2A6CYP2E1CYP3A4CYP2D6CYP2C9
SCHEMBL9988058 0.77 CYP2C9 (0.40) CYP2A6CYP2E1CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL1156993 0.77 CYP2E1 (0.39) CYP2A6CYP2E1CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919865-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2008-05-14 EP disclosed
WO-2007026916-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-03-08 WO disclosed