SCHEMBL4792177

SCHEMBL4792177

C[C](c1cc(-c2ncccc2C)n(S(=O)(=O)c2cccnc2)c1)C(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.37
CHRM5 P08912 1/20 0.36
RAPGEF4 Q8WZA2 2/20 0.35
GPBAR1 Q8TDU6 1/20 0.35
MET P08581 5/20 0.34
NAPRT Q6XQN6 1/20 0.34
PTGS2 P35354 2/20 0.33
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
POLB P06746 1/20 0.33
KMT2A Q03164 1/20 0.33
SMO Q99835 1/20 0.33
KDM4E B2RXH2 1/20 0.33
SLC40A1 Q9NP59 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4793151 0.85 PTGES2 (0.35) CHRM5NAPRTPTGS2MAPTSMN1; SMN2
SCHEMBL4790340 0.82 CYP2A6 (0.42) CYP2A6CHRM5NAPRTMAPTSMN1; SMN2
SCHEMBL4793065 0.80 PTGS2 (0.44) PTGS2
SCHEMBL4791372 0.80 GBA1 (0.40) CYP2A6NAPRTMAPTSMN1; SMN2POLB
SCHEMBL4792179 0.79 CYP2A6 (0.36) CYP2A6CHRM5RAPGEF4METPTGS2
SCHEMBL1581058 0.76 TSHR (0.38) CYP2A6CHRM5RAPGEF4METMAPT
SCHEMBL9988642 0.76 TSHR (0.41) KMT2A
SCHEMBL1278610 0.74 RIPK1 (0.34) CHRM5GPBAR1MAPTSMN1; SMN2
Fumaric Acid SCHEMBL1278719 0.72 HDAC1 (0.35) SMN1; SMN2POLBKMT2AKDM4E
Fumaric Acid SCHEMBL1278717 0.72 HDAC1 (0.35) SMN1; SMN2POLBKMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919865-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2008-05-14 EP disclosed
WO-2007026916-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-03-08 WO disclosed