SCHEMBL4791682

SCHEMBL4791682

COc1ccc(C)cc1-c1cc(F)cc2c1O[CH]C2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.37
ALDH1A1 P00352 3/20 0.34
CYP3A4 P08684 1/20 0.34
CTSA P10619 2/20 0.34
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
LMNA P02545 3/20 0.33
CCNT1 O60563 3/20 0.32
CDK9 P50750 3/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
KDM4E B2RXH2 1/20 0.32
MDM2 Q00987 1/20 0.32
DHODH Q02127 1/20 0.32
LRRK2 Q5S007 1/20 0.31
RPS6KA2 Q15349 1/20 0.31
USP2 O75604 1/20 0.31
GAA P10253 1/20 0.31
KMT2A Q03164 1/20 0.31
MAPT P10636 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27703038 0.84 HTR7 (0.38) ALDH1A1CYP3A4HTR2AHTR2CLMNA
SCHEMBL4608823 0.78 NFE2L2 (0.36) ALDH1A1HTR2AHTR2CLMNASMN1; SMN2
SCHEMBL4595097 0.77 PARP1 (0.43) ACHEALDH1A1CCNT1CDK9SMN1; SMN2
SCHEMBL27703250 0.77 HTR7 (0.39) ALDH1A1CYP3A4SMN1; SMN2KDM4EUSP2
SCHEMBL4595096 0.76 AQP1 (0.35) ACHEALDH1A1CYP3A4CTSAHTR2A
SCHEMBL4760683 0.75 CA12 (0.41) ALDH1A1LMNASMN1; SMN2KDM4EGAA
SCHEMBL27703115 0.74 MAPT (0.39) MAPTBACE1
SCHEMBL5137212 0.74 HTR2A (0.42) ALDH1A1HTR2AHTR2CSMN1; SMN2KDM4E
SCHEMBL4220657 0.73 AQP1 (0.56) HTR2C
SCHEMBL4220133 0.72 AQP1 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1898895-A2 TREATMENT OF DRUG ABUSE Wyeth (US) 2008-03-19 EP disclosed
EP-1871356-A1 DIHYDROBENZOFURAN DERIVATIVES AND USES THEREOF Wyeth a Corporation of the State of Delaware (US) 2008-01-02 EP disclosed
WO-2006116170-A1 DIHYDROBENZOFURAN DERIVATIVES AND USES THEREOF WYETH (US) 2006-11-02 WO disclosed
WO-2006116148-A2 (7-ARLYSUBSTITUTED 2, 3-DIHYDR0-1-BENZ0FURAN-2-YL) ALKYLAMINES IN THE TREATMENT' OF SUBSTANCE ABUSE WYETH (US) 2006-11-02 WO disclosed