SCHEMBL4792118

SCHEMBL4792118

OCc1nn(-c2ccc(Cl)cc2)c2ccccc12

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RORC P51449 6/20 0.51
RARG P13631 4/20 0.51
NOTUM Q6P988 1/20 0.48
PDE5A O76074 1/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
GAA P10253 1/20 0.43
PTGS1 P23219 1/20 0.43
PTGS2 P35354 1/20 0.43
ABCB1 P08183 5/20 0.41
TEAD1 P28347 1/20 0.41
TEAD4 Q15561 1/20 0.41
TEAD2 Q15562 1/20 0.41
TEAD3 Q99594 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27834343 0.87 PDE5A (0.55) RORCRARGPDE5ASMN1; SMN2TEAD1
SCHEMBL4793748 0.86 RORC (0.49) RORCRARGNPC1RAB9ASMN1; SMN2
SCHEMBL4792507 0.81 MAPT (0.47) RORCRARGNOTUMPDE5ARAB9A
SCHEMBL928140 0.80 PTGER4 (0.50) PDE5ANPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL3157520 0.79 RORC (0.47) RORCRARGNPC1RAB9ASMN1; SMN2
SCHEMBL4792952 0.77 TEAD1 (0.63) RORCRARGPDE5AABCB1TEAD1
SCHEMBL12253498 0.76 GAA (0.67) NPC1RAB9ASMN1; SMN2GAAALDH1A1
SCHEMBL3347837 0.74 L3MBTL1 (0.38) RORCRARGPDE5ANPC1RAB9A
SCHEMBL4792972 0.74 SCN9A (0.42) NOTUMPTGS1PTGS2
SCHEMBL4795769 0.74 EGLN2 (0.41) NOTUMPTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937647-A1 CONDENSED PYRAZOLE DERIVATIVES AS PPAR AGONISTS II Inpharmatica Limited (GB) 2008-07-02 EP disclosed
WO-2007036727-A1 CONDENSED PYRAZOLE DERIVATIVES AS PPAR AGONISTS II INPHARMATICA LIMITED (GB) 2007-04-05 WO disclosed
WO-2007036727-A1 CONDENSED PYRAZOLE DERIVATIVES AS PPAR AGONISTS II INPHARMATICA LIMITED (GB) 2007-04-05 WO disclosed