SCHEMBL4794017

SCHEMBL4794017

O=Cc1ccc(C(=O)NN(C(=O)O)c2ccc(-c3cccs3)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC2 Q92769 3/20 0.44
HPGDS O60760 1/20 0.42
HDAC1 Q13547 7/20 0.40
HDAC3 O15379 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
TNFRSF1A P19438 1/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
KMT2A Q03164 1/20 0.39
ERN1 O75460 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
DRD2 P14416 3/20 0.38
DRD4 P21917 3/20 0.38
HTR2A P28223 1/20 0.38
ABL1 P00519 2/20 0.37
BCR P11274 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1066552 0.86 ABL1 (0.52) HDAC2HPGDSHDAC1HDAC3L3MBTL1
SCHEMBL2464650 0.84 HDAC2 (0.60) HDAC2HDAC1HDAC3TNFRSF1AKDM4E
SCHEMBL2685210 0.84 GPR119 (0.43) HDAC2HPGDSHDAC1HDAC3L3MBTL1
SCHEMBL4669170 0.84 HDAC1 (0.48) HPGDSHDAC1DRD2DRD4HTR2A
SCHEMBL4579392 0.83 HPGDS (0.46) HPGDSHDAC1DRD2DRD4HTR2A
SCHEMBL4580709 0.79 TDP1 (0.51) HDAC2HPGDSHDAC1HDAC3L3MBTL1
SCHEMBL4579334 0.77 HPGDS (0.40) HDAC2HPGDSHDAC1HDAC3L3MBTL1
SCHEMBL1068512 0.76 ABL1 (0.54) HDAC2HDAC1HDAC3L3MBTL1KDM4E
SCHEMBL29898509 0.75 HDAC2 (0.48) HDAC2HDAC1HDAC3TNFRSF1AKDM4E
SCHEMBL29898510 0.75 HDAC2 (0.48) HDAC2HDAC1HDAC3TNFRSF1AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1991226-A2 INHIBITORS OF HISTONE DEACETYLASE Merck & Co., Inc. (US) 2008-11-19 EP disclosed
WO-2007100657-A2 INHIBITORS OF HISTONE DEACETYLASE MERCK & CO., INC. (US) 2007-09-07 WO disclosed