SCHEMBL4795580

SCHEMBL4795580

Cc1cc(N)nc2c1CN(c1ccc(F)cc1)C=C2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.36
KMT2A Q03164 4/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35
NOS2 P35228 1/20 0.35
KDM4E B2RXH2 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
LMNA P02545 2/20 0.32
DHFR P00374 1/20 0.32
RXRA P19793 1/20 0.31
GRIN1 Q05586 1/20 0.31
GRIN2B Q13224 1/20 0.31
MAPT P10636 2/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPK1 P28482 1/20 0.30
HTT P42858 1/20 0.30
GFER P55789 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4796617 0.84 DHFR (0.34) SMN1; SMN2DHFRCYP3A4DPP4DPP8
SCHEMBL4759492 0.81 MCHR1 (0.33)
SCHEMBL5814749 0.61 ADORA2A (0.35) MEN1KMT2ANPC1RAB9AKDM4E
SCHEMBL25070257 0.59 ALDH1A1 (0.40) NPC1RAB9AKDM4ELMNADHFR
SCHEMBL4129260 0.57
SCHEMBL27710876 0.57 PARP1 (0.34) MEN1KMT2ANPC1RAB9AKDM4E
SCHEMBL14749859 0.56 NPC1 (0.50) MEN1KMT2ANPC1RAB9AKDM4E
SCHEMBL20414976 0.56 ALDH1A1 (0.41) MEN1KMT2ANPC1RAB9AKDM4E
SCHEMBL4782650 0.55
SCHEMBL5741120 0.55 HRH4 (0.59) MEN1KMT2ANPC1RAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009076-A2 SUBSTITUTED PYRIDO(3,2-D)PYRIMIDINES AND PHARMACEUTICAL COMPOSITIONS FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-01-24 WO claimed