SCHEMBL4796617

SCHEMBL4796617

CCc1cc(N)nc2c1CN(c1ccc(F)cc1)C=C2

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DHFR P00374 2/20 0.34
MPO P05164 5/20 0.32
CYP3A4 P08684 2/20 0.32
TPO P07202 1/20 0.32
KCNH2 Q12809 1/20 0.31
PDE4A P27815 3/20 0.31
PDE4B Q07343 3/20 0.31
PDE4C Q08493 3/20 0.31
PDE4D Q08499 3/20 0.31
DPP4 P27487 1/20 0.31
DPP8 Q6V1X1 1/20 0.31
DPP9 Q86TI2 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4795580 0.84 MEN1 (0.36) DHFRCYP3A4DPP4DPP8DPP9
SCHEMBL4794363 0.82 ALDH1A1 (0.37) SMN1; SMN2
SCHEMBL4759492 0.78 MCHR1 (0.33) KCNH2
SCHEMBL4796924 0.72 MEN1 (0.34) SMN1; SMN2
SCHEMBL4790457 0.61 TLR8 (0.38) MPOKCNH2SMN1; SMN2
SCHEMBL25070257 0.57 ALDH1A1 (0.40) DHFR
SCHEMBL17236140 0.56 NOS2 (0.42) MPO
SCHEMBL18315118 0.55 NOS2 (0.45)
Hydrochloric Acid SCHEMBL17224997 0.55 NOS2 (0.41) MPO
SCHEMBL4129260 0.55

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009076-A2 SUBSTITUTED PYRIDO(3,2-D)PYRIMIDINES AND PHARMACEUTICAL COMPOSITIONS FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-01-24 WO disclosed