SCHEMBL4797150

SCHEMBL4797150

CC(C)CC1(C(=O)NCc2cc(C(F)(F)F)cc(C(F)(F)F)c2)CCNCC1

nearest known ligand 0.59

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.59
CCR2 P41597 17/20 0.49
CYP3A4 P08684 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL3038763 0.96 TACR1 (0.58) TACR1CCR2CYP3A4
SCHEMBL5728946 0.82 CCR2 (0.50) TACR1CCR2CYP3A4
SCHEMBL14221691 0.82 TACR1 (0.65) TACR1CCR2CYP3A4
SCHEMBL3029909 0.81 TACR1 (0.59) TACR1CCR2
SCHEMBL3029890 0.81 CCR2 (0.51) CCR2CYP3A4
Ammonia Solution, Strong SCHEMBL3036646 0.81 TACR1 (0.64) TACR1CCR2CYP3A4
SCHEMBL3038764 0.80 CCR2 (0.48) CCR2CYP3A4
SCHEMBL7919481 0.79 ATM (0.53) TACR1
SCHEMBL4731356 0.78 TACR1 (0.44) TACR1CCR2CYP3A4
Trifluoroacetic Acid SCHEMBL3030594 0.78 TACR1 (0.64) TACR1CCR2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008045564-A2 CARBOXAMIDE COMPOUNDS AND THEIR USE AS ANTAGONISTS OF THE CHEMOKINE CCR2 RECEPTOR EPIX DELAWARE, INC. (US) 2008-04-17 WO disclosed