SCHEMBL480055

SCHEMBL480055

COC(=O)c1ccc(-c2ccc(C(C)C(O)(c3ccnc(-c4ccc(C(=O)O)cc4)c3)C(F)(F)F)cc2)c(C(C)C(O)(c2ccnc(-c3ccc(C(=O)O)cc3)c2)C(F)(F)F)c1Cl

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.35
CYP2C8 P10632 2/20 0.34
LOXL2 Q9Y4K0 1/20 0.34
PTGER4 P35408 4/20 0.33
BDKRB1 P46663 2/20 0.33
KDM4E B2RXH2 1/20 0.33
KDM6B O15054 1/20 0.33
KDM5C P41229 1/20 0.33
KDM4C Q9H3R0 1/20 0.33
KDM2A Q9Y2K7 1/20 0.33
KDM3A Q9Y4C1 1/20 0.33
KMO O15229 1/20 0.32
AKR1C3 P42330 2/20 0.32
AKR1C2 P52895 2/20 0.32
SRD5A2 P31213 2/20 0.32
ROCK2 O75116 1/20 0.31
ROCK1 Q13464 1/20 0.31
PTGER2 P43116 1/20 0.31
TGFBR1 P36897 1/20 0.31
CCNT1 O60563 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL480056 0.83 BDKRB1 (0.42) PTGER4BDKRB1KMO
SCHEMBL733519 0.81 SLC6A3 (0.39) PDK2PTGER4BDKRB1KDM4EKDM6B
SCHEMBL733518 0.80 KDM4E (0.39) PDK2LOXL2KDM4EKDM6BKDM5C
SCHEMBL480017 0.79 KDM4E (0.39) PDK2LOXL2KDM4EKDM6BKDM5C
SCHEMBL754770 0.76 KMO (0.43) PDK2LOXL2KDM4CKMO
SCHEMBL479917 0.76 KMO (0.43) PDK2LOXL2KDM4CKMO
SCHEMBL837203 0.74 CHEK1 (0.39) CYP2C8LOXL2KDM4EKDM4CKMO
SCHEMBL15789725 0.72 KMO (0.38) LOXL2KDM4CKMOSRD5A2
SCHEMBL480633 0.69 SLC6A3 (0.42) PDK2BDKRB1ROCK2ROCK1
SCHEMBL755473 0.68 ROCK2 (0.39) PDK2KDM4EROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed