SCHEMBL480164

SCHEMBL480164

C[C@H](Cl)OC(=O)c1ccc(B(O)O)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 4/20 0.46
CA1 P00915 3/20 0.46
CA12 O43570 2/20 0.46
CA7 P43166 2/20 0.46
CA9 Q16790 2/20 0.46
CA14 Q9ULX7 2/20 0.46
PDCD1 Q15116 1/20 0.42
CD274 Q9NZQ7 1/20 0.42
CYP4F2 P78329 1/20 0.40
CYP4A11 Q02928 1/20 0.40
ENPP2 Q13822 3/20 0.38
LPL P06858 2/20 0.38
LIPG Q9Y5X9 2/20 0.38
ALDH1A1 P00352 3/20 0.38
TRPV1 Q8NER1 2/20 0.37
NPC1 O15118 1/20 0.37
LMNA P02545 1/20 0.37
HTT P42858 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL141580 0.85 CA12 (0.63) CA2CA1CA12CA7CA9
SCHEMBL11058125 0.79 CA12 (0.71) CA2CA1CA12CA7CA9
SCHEMBL5672629 0.77 TSHR (0.59) CA2CA1CA12CA7CA9
SCHEMBL27610990 0.77 TSHR (0.59) CA2CA1CA12CA7CA9
SCHEMBL1594032 0.77 TSHR (0.59) CA2CA1CA12CA7CA9
SCHEMBL11478296 0.76 CA1 (0.60) CA2CA1CA12CA7CA9
SCHEMBL140644 0.75 CA1 (0.59) CA2CA1CA12CA7CA9
SCHEMBL26901115 0.74 ALDH1A1 (0.51) ALDH1A1NPC1HTTRAB9A
SCHEMBL2040977 0.73 CA1 (0.57) CA2CA1CA12CA7CA9
SCHEMBL28754539 0.72 ALDH1A1 (0.53) CA2CA1ALDH1A1NPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed