SCHEMBL480182

SCHEMBL480182

Cc1[nH]c(=O)ccc1C(O)(C(C)c1ccc(-c2ccc(C(=O)O)c(F)c2)cc1Cl)C(F)(F)F

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.33
RARB P10826 4/20 0.33
RARA P10276 3/20 0.33
RARG P13631 2/20 0.33
PRKAB2 O43741 1/20 0.33
PRKAG1 P54619 1/20 0.33
PRKAA2 P54646 1/20 0.33
PRKAA1 Q13131 1/20 0.33
PRKAG3 Q9UGI9 1/20 0.33
PRKAG2 Q9UGJ0 1/20 0.33
PRKAB1 Q9Y478 1/20 0.33
ADRA2A P08913 1/20 0.32
CLCN2 P51788 1/20 0.32
RORC P51449 1/20 0.32
SCN5A Q14524 1/20 0.31
PDE2A O00408 4/20 0.31
RXRA P19793 1/20 0.31
RXRB P28702 1/20 0.31
DHODH Q02127 1/20 0.31
PDK2 Q15119 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL480109 0.93 PDK2 (0.36) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL480166 0.90 BDKRB1 (0.36) SCN9ASCN5APDE2APDK2NPC1
SCHEMBL479986 0.88 PRKAB2 (0.37) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL480185 0.85 PDK2 (0.40) PDE2APDK2
SCHEMBL480320 0.83 SCN9A (0.34) SCN9A
SCHEMBL752284 0.82 PRKAB2 (0.34) RARBRARARARGPRKAB2PRKAG1
SCHEMBL480080 0.82 PRKAB2 (0.34) RARBRARARARGPRKAB2PRKAG1
SCHEMBL480086 0.82 CHEK1 (0.37) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL480013 0.80 RXRB (0.35) RARBRARARARGPRKAB2PRKAG1
SCHEMBL12187886 0.79 GRIA1 (0.38) RARBRARARARGPRKAB2PRKAG1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP claimed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO claimed