SCHEMBL480320

SCHEMBL480320

Cc1[nH]c(=O)ccc1C(O)(C(C)c1cc(F)c(Oc2ccc(C(=O)O)c(F)c2)cc1Cl)C(F)(F)F

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 7/20 0.34
SCN8A Q9UQD0 4/20 0.34
SCN10A Q9Y5Y9 4/20 0.34
RHEB Q15382 1/20 0.32
GPR35 Q9HC97 1/20 0.31
MEN1 O00255 1/20 0.30
TTR P02766 1/20 0.30
PPOX P50336 1/20 0.30
KMT2A Q03164 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL480155 0.92 SCN8A (0.36) SCN9ASCN8ASCN10A
SCHEMBL480084 0.84 S1PR2 (0.33) RHEB
SCHEMBL479955 0.83 IGFBP3 (0.35) RHEB
SCHEMBL480182 0.83 SCN9A (0.33) SCN9A
SCHEMBL480037 0.82 SCN8A (0.34) SCN9ASCN8ASCN10ARHEBMEN1
SCHEMBL15789678 0.80 MCL1 (0.35) RHEB
SCHEMBL754534 0.79 SCN8A (0.35) SCN9ASCN8ASCN10AMEN1TTR
SCHEMBL733289 0.79 SCN8A (0.35) SCN9ASCN8ASCN10AMEN1TTR
SCHEMBL480109 0.78 PDK2 (0.36)
SCHEMBL480171 0.78 CYP11B1 (0.35) SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP claimed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO claimed