SCHEMBL480013

SCHEMBL480013

Cc1cc(C(O)(C(C)c2ccc(-c3ccc(C(=O)O)c(F)c3)cc2Cl)C(F)(F)F)c[nH]c1=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRB P28702 2/20 0.35
RXRA P19793 1/20 0.35
ERCC1 P07992 1/20 0.34
ERCC4 Q92889 1/20 0.34
ADRA2A P08913 1/20 0.34
CLCN2 P51788 1/20 0.34
PRKAB2 O43741 3/20 0.33
PRKAG1 P54619 3/20 0.33
PRKAA2 P54646 3/20 0.33
PRKAA1 Q13131 3/20 0.33
PRKAG3 Q9UGI9 3/20 0.33
PRKAG2 Q9UGJ0 3/20 0.33
PRKAB1 Q9Y478 3/20 0.33
RARB P10826 4/20 0.33
RARA P10276 3/20 0.33
RARG P13631 2/20 0.33
PIK3CG P48736 1/20 0.33
RET P07949 2/20 0.31
AXL P30530 1/20 0.31
ADRB2 P07550 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL479731 0.93 RXRB (0.37) RXRBRXRAERCC1ERCC4ADRA2A
SCHEMBL479948 0.93 ERCC1 (0.36) RXRBRXRAERCC1ERCC4ADRA2A
SCHEMBL480103 0.91 GRIK1 (0.40) RXRBRXRAERCC1ERCC4ADRA2A
SCHEMBL479738 0.90 BDKRB1 (0.35) ERCC1ERCC4RETPDK2
SCHEMBL480032 0.90 RARB (0.35) ERCC1ERCC4PRKAB2PRKAG1PRKAA2
SCHEMBL480020 0.88 PRKAB2 (0.33) ADRA2ACLCN2PRKAB2PRKAG1PRKAA2
SCHEMBL480183 0.88 PRKAB2 (0.37) RXRBRXRAPRKAB2PRKAG1PRKAA2
SCHEMBL752284 0.88 PRKAB2 (0.34) RXRBRXRAERCC1ERCC4PRKAB2
SCHEMBL480080 0.88 PRKAB2 (0.34) RXRBRXRAERCC1ERCC4PRKAB2
SCHEMBL479944 0.85 RXRA (0.39) RXRBRXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed