SCHEMBL480204

SCHEMBL480204

CCOC(=O)c1cc(-c2ccc(C(C)C(O)(c3c[nH]c(=O)c(C)c3)C(F)(F)F)c(Cl)c2)ccc1F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 2/20 0.34
ERCC1 P07992 1/20 0.34
ERCC4 Q92889 1/20 0.34
MRGPRX4 Q96LA9 1/20 0.34
NPC1 O15118 1/20 0.34
RET P07949 2/20 0.34
PTPRC P08575 1/20 0.34
PTPN2 P17706 1/20 0.34
PTPN1 P18031 1/20 0.34
PTPA Q15257 1/20 0.34
KDM4E B2RXH2 3/20 0.33
TEAD2 Q15562 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
JAK2 O60674 1/20 0.33
JAK3 P52333 1/20 0.33
BAZ2B Q9UIF8 1/20 0.32
BAZ2A Q9UIF9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL479902 0.93 MRGPRX4 (0.35) BDKRB1ERCC1ERCC4MRGPRX4NPC1
SCHEMBL479948 0.89 ERCC1 (0.36) ERCC1ERCC4MRGPRX4
SCHEMBL479738 0.85 BDKRB1 (0.35) BDKRB1ERCC1ERCC4NPC1RET
SCHEMBL479871 0.85 MRGPRX4 (0.33) MRGPRX4KDM4ENPSR1HPGDMEN1
SCHEMBL480013 0.84 RXRB (0.35) ERCC1ERCC4RET
SCHEMBL480079 0.84 PDK2 (0.40) BDKRB1ERCC1ERCC4ALDH1A1HPGD
SCHEMBL480103 0.84 GRIK1 (0.40) ERCC1ERCC4ALDH1A1GAAMAPT
SCHEMBL480005 0.83 ERCC1 (0.35) ERCC1ERCC4MRGPRX4RETPTPRC
SCHEMBL479731 0.83 RXRB (0.37) ERCC1ERCC4SMN1; SMN2
SCHEMBL754461 0.82 BAZ2B (0.44) BDKRB1MRGPRX4NPC1PTPRCPTPN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed