SCHEMBL480079

SCHEMBL480079

COC(=O)c1ccc(-c2ccc(C(C)C(O)(c3c[nH]c(=O)c(C)c3)C(F)(F)F)c(Cl)c2)cc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.40
ACLY P53396 1/20 0.36
BDKRB1 P46663 2/20 0.32
CFTR P13569 1/20 0.31
ROCK2 O75116 1/20 0.31
ROCK1 Q13464 1/20 0.31
NR4A2 P43354 5/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
ALOX12 P18054 1/20 0.31
MAPK1 P28482 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
PDE2A O00408 1/20 0.31
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31
ERCC1 P07992 1/20 0.30
ERCC4 Q92889 1/20 0.30
P2RX3 P56373 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL479738 0.94 BDKRB1 (0.35) PDK2ACLYBDKRB1ERCC1ERCC4
SCHEMBL480057 0.93 CHEK1 (0.37) PDK2ACLYROCK2ROCK1ALDH1A1
SCHEMBL479964 0.91 KDR (0.32) PDK2ACLYCFTRALDH1A1LMNA
SCHEMBL479731 0.90 RXRB (0.37) PDK2SMN1; SMN2PDE2AERCC1ERCC4
SCHEMBL480183 0.86 PRKAB2 (0.37) ROCK2ROCK1ALDH1A1
SCHEMBL480013 0.85 RXRB (0.35) PDK2ERCC1ERCC4
SCHEMBL480103 0.85 GRIK1 (0.40) PDK2ALDH1A1MAPTERCC1ERCC4
SCHEMBL479739 0.85 KDR (0.33) PDK2MAPT
SCHEMBL480130 0.84 RET (0.37) PDK2ACLYBDKRB1
SCHEMBL480204 0.84 BDKRB1 (0.34) BDKRB1ALDH1A1MAPTHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed