SCHEMBL479738

SCHEMBL479738

COC(=O)c1ccc(-c2ccc(C(C)C(O)(c3c[nH]c(=O)c(C)c3)C(F)(F)F)c(Cl)c2)cc1F

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 6/20 0.35
PDK2 Q15119 1/20 0.35
ACLY P53396 1/20 0.35
RET P07949 5/20 0.33
MET P08581 4/20 0.33
ERCC1 P07992 1/20 0.33
ERCC4 Q92889 1/20 0.33
NPC1 O15118 1/20 0.33
SCN5A Q14524 1/20 0.32
SCN9A Q15858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL480079 0.94 PDK2 (0.40) BDKRB1PDK2ACLYERCC1ERCC4
SCHEMBL480130 0.91 RET (0.37) BDKRB1PDK2ACLYRETNPC1
SCHEMBL480057 0.90 CHEK1 (0.37) PDK2ACLYRET
SCHEMBL480013 0.90 RXRB (0.35) PDK2RETERCC1ERCC4
SCHEMBL479731 0.85 RXRB (0.37) PDK2ERCC1ERCC4
SCHEMBL480204 0.85 BDKRB1 (0.34) BDKRB1RETERCC1ERCC4NPC1
SCHEMBL479964 0.85 KDR (0.32) PDK2ACLY
SCHEMBL479948 0.85 ERCC1 (0.36) ERCC1ERCC4
SCHEMBL479721 0.84 P2RX3 (0.34) METSCN5ASCN9A
SCHEMBL480183 0.84 PRKAB2 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed