SCHEMBL4802137

SCHEMBL4802137

O=C1NNC([Pt])c2ccccc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.39
HTR2C P28335 2/20 0.39
HTR2B P41595 2/20 0.39
PARP1 P09874 1/20 0.39
GSK3B P49841 1/20 0.38
HSD17B10 Q99714 2/20 0.38
PARP3 Q9Y6F1 1/20 0.36
EDNRB P24530 1/20 0.35
EDNRA P25101 1/20 0.35
TNKS2 Q9H2K2 3/20 0.35
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PBRM1 Q86U86 1/20 0.35
CASP3 P42574 1/20 0.33
CASP2 P42575 1/20 0.33
CASP7 P55210 1/20 0.33
CASP6 P55212 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19675124 0.76 S100A4 (0.40) HTR2AHTR2CHTR2BPARP1GSK3B
SCHEMBL19675259 0.71 PARP3 (0.39) HTR2AHTR2CHTR2BPARP1GSK3B
SCHEMBL10517286 0.67 HSD17B10 (0.51) HSD17B10PARP3EDNRBEDNRATSHR
SCHEMBL5009457 0.66 HTR2C (0.42) HTR2AHTR2CHTR2BPARP1PARP3
Zinc Ion SCHEMBL10517280 0.66 HSD17B10 (0.50) HTR2AHTR2CHTR2BPARP1HSD17B10
SCHEMBL1443391 0.64 TNKS2 (0.52) HTR2AHTR2CHTR2BPARP1HSD17B10
SCHEMBL24038969 0.63 HTR2A (0.67) HTR2AHTR2CHTR2BPARP1GSK3B
SCHEMBL19696037 0.63 HTR2A (0.67) HTR2AHTR2CHTR2BPARP1GSK3B
SCHEMBL19696047 0.63 HTR2A (0.67) HTR2AHTR2CHTR2BPARP1GSK3B
SCHEMBL4914352 0.63 HSD17B10 (0.51) HTR2AHTR2CHTR2BPARP1GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1896491-A2 MONOAZOLE LIGAND PLATINUM ANALOGS BIONUMERIK PHARMACEUTICALS, INC. (US) 2008-03-12 EP disclosed
WO-2007005058-A2 MONOAZOLE LIGAND PLATINUM ANALOGS BIONUMERIK PHARMACEUTICALS, INC. (US) 2007-01-11 WO disclosed