SCHEMBL19675259

SCHEMBL19675259

Nc1ccc(C2NNC(=O)c3ccccc32)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP3 Q9Y6F1 1/20 0.39
HTR2A P28223 2/20 0.38
HTR2C P28335 2/20 0.38
HTR2B P41595 2/20 0.38
PARP1 P09874 1/20 0.38
CYP19A1 P11511 1/20 0.38
JAK2 O60674 1/20 0.37
HSD17B10 Q99714 1/20 0.37
AKT1 P31749 1/20 0.36
DDB1 Q16531 1/20 0.36
CRBN Q96SW2 1/20 0.36
GSK3B P49841 1/20 0.36
NPC1 O15118 2/20 0.35
ALDH1A1 P00352 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
TP53 P04637 1/20 0.35
CYP3A4 P08684 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19675594 0.80 CYP26A1 (0.39) CYP19A1HSD17B10DDB1CRBNALDH1A1
SCHEMBL19675765 0.76 ALDH1A1 (0.38) HTR2AHTR2CHTR2BPARP1HSD17B10
SCHEMBL19675735 0.73 HSD17B10 (0.37) PARP3HTR2AHTR2CHTR2BPARP1
SCHEMBL19675124 0.71 S100A4 (0.40) PARP3HTR2AHTR2CHTR2BPARP1
SCHEMBL1443391 0.71 TNKS2 (0.52) PARP3HTR2AHTR2CHTR2BPARP1
SCHEMBL4802137 0.71 HTR2A (0.39) PARP3HTR2AHTR2CHTR2BPARP1
SCHEMBL1444438 0.69 ALDH1A1 (0.57) HTR2AHTR2CHTR2BPARP1HSD17B10
SCHEMBL29155427 0.69 SMN1; SMN2 (0.58) PARP3HTR2AHTR2CHTR2BPARP1
SCHEMBL30683790 0.69 SMN1; SMN2 (0.58) PARP3HTR2AHTR2CHTR2BPARP1
SCHEMBL29506922 0.69 TNKS2 (0.57) HTR2AHTR2CHTR2BPARP1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3252049-A1 PHTHALAZINONES AND ISOQUINOLINONES AS ROCK INHIBITORS Bristol-Myers Squibb Company (US) 2017-12-06 EP disclosed
EP-3252050-A1 PHTHALAZINONES AND ISOQUINOLINONES AS ROCK INHIBITORS Bristol-Myers Squibb Company (US) 2017-12-06 EP disclosed