SCHEMBL4806740

SCHEMBL4806740

CC(=O)[C@](I)(Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 4/20 0.52
CTSL P07711 2/20 0.52
CTSS P25774 1/20 0.52
CTSK P43235 1/20 0.52
MAPT P10636 4/20 0.49
TP53 P04637 1/20 0.49
SSTR3 P32745 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
ACE P12821 1/20 0.47
P4HB P07237 4/20 0.46
GAA P10253 3/20 0.46
POLB P06746 1/20 0.46
TSHR P16473 2/20 0.45
LMNA P02545 1/20 0.45
CYP1A2 P05177 1/20 0.45
PKM P14618 1/20 0.45
CYP2C19 P33261 1/20 0.45
BLM P54132 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3020291 0.81 CTSL (0.59) TACR1CTSLCTSSCTSKMAPT
SCHEMBL3020294 0.81 CTSL (0.59) TACR1CTSLCTSSCTSKMAPT
SCHEMBL9016089 0.81 CTSL (0.59) TACR1CTSLCTSSCTSKMAPT
SCHEMBL8651829 0.81 CTSL (0.58) TACR1CTSLCTSSCTSKMAPT
SCHEMBL2193454 0.81 CTSL (0.55) TACR1CTSLCTSSCTSKMAPT
SCHEMBL8650748 0.80 CTSL (0.57) TACR1CTSLCTSSCTSKMAPT
SCHEMBL9270557 0.78 CTSL (0.55) TACR1CTSLCTSSCTSKMAPT
SCHEMBL8650822 0.77 CTSL (0.62) TACR1CTSLCTSSCTSKMAPT
SCHEMBL19100705 0.77 CTSL (0.58) TACR1CTSLCTSSCTSKMAPT
SCHEMBL24178475 0.76 CTSL (0.67) TACR1CTSLCTSSCTSKMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008071453-A1 1,2-DIARYLACETYLENE DERIVATIVES OF ACYLTRYPTOPHANOLS BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2008-06-19 WO disclosed