SCHEMBL4819508

SCHEMBL4819508

[CH2]c1ccc(OCCO)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.60
RECQL P46063 1/20 0.60
NR1I2 O75469 1/20 0.53
GAA P10253 1/20 0.50
CYP3A4 P08684 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
APP P05067 5/20 0.42
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA9 Q16790 1/20 0.41
ALOX5AP P20292 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CYP19A1 P11511 1/20 0.39
PRSS1 P07477 1/20 0.39
MEN1 O00255 1/20 0.39
USP2 O75604 1/20 0.39
LMNA P02545 1/20 0.39
MAPK1 P28482 1/20 0.39
CASP1 P29466 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28106819 0.87 ALDH1A1 (0.75) ALDH1A1RECQLNR1I2GAACYP3A4
SCHEMBL48239 0.87 ALDH1A1 (0.75) ALDH1A1RECQLNR1I2GAACYP3A4
Ethylene Glycol SCHEMBL11119213 0.85 ALDH1A1 (0.71) ALDH1A1RECQLNR1I2GAACYP3A4
Water SCHEMBL29229746 0.85 ALDH1A1 (0.71) ALDH1A1RECQLNR1I2GAACYP3A4
SCHEMBL8019585 0.85 PRMT1 (0.46) ALDH1A1RECQLGAAL3MBTL1PRSS1
SCHEMBL2720663 0.82 ALDH1A1 (0.68) ALDH1A1RECQLNR1I2GAACYP3A4
SCHEMBL9119081 0.82 ALDH1A1 (0.68) ALDH1A1RECQLNR1I2GAACYP3A4
SCHEMBL14004241 0.82 ALDH1A1 (0.68) ALDH1A1RECQLNR1I2GAACYP3A4
SCHEMBL152501 0.82 ALDH1A1 (0.68) ALDH1A1RECQLNR1I2GAACYP3A4
SCHEMBL14151809 0.82 ALDH1A1 (0.56) ALDH1A1RECQLNR1I2GAACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE37781-E1 VIRICIDES, PROTEASE INHIBITOR DUPONT PHARMACEUTICALS COMPANY 2002-07-02 US claimed
US-5811422-A USEFUL FOR TREATING VIRAL INFECTIONS THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1998-09-22 US claimed
US-5710286-A Processes and intermediates for the preparation of cyclic urea HIV protease inhibitors THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1998-01-20 US claimed
US-5610294-A VIRAL TREATMENT THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-03-11 US claimed
US-5559110-A HIV ANTIVIRAL, GOOD SYSTEMIC ABSORPTION ADMINISTERED BY MOUTH THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1996-09-24 US claimed
WO-1996000728-A1 PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF CYCLIC UREA HIV PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-01-11 WO claimed
EP-0686151-A1 SUBSTITUTED CYCLIC CARBONYLS AND DERIVATIVES THEREOF USEFUL AS RETROVIRAL PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-12-13 EP claimed
US-5466797-A Intermediates for the preparation of cyclic urea THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-11-14 US claimed
WO-1994019329-A1 SUBSTITUTED CYCLIC CARBONYLS AND DERIVATIVES THEREOF USEFUL AS RETROVIRAL PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1994-09-01 WO claimed
US-7402696-B2 Benzene compounds AJINOMOTO CO., INC. (JP) 2008-07-22 US disclosed
US-20070105899-A1 Benzene compounds AJINOMOTO CO., INC. (JP) 2007-05-10 US disclosed
US-6503898-B1 Administering 4,7-dibenzyl-5,6-dihydroxy-N,N*-di(m-aminobenzyl)--1,3-diazepin-2-one or salt to treat human immunodeficiency virus infection BRISTOL-MYERS SQUIBB PHARMA COMPANY 2003-01-07 US disclosed
US-RE37781-E1 VIRICIDES, PROTEASE INHIBITOR DUPONT PHARMACEUTICALS COMPANY 2002-07-02 US disclosed
US-6054597-A Processes and intermediates for the preparation of cyclic urea HIV protease inhibitors DUPONT PHARMACEUTICALS (US) 2000-04-25 US disclosed
US-5610294-A VIRAL TREATMENT THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-03-11 US disclosed
US-5559110-A HIV ANTIVIRAL, GOOD SYSTEMIC ABSORPTION ADMINISTERED BY MOUTH THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1996-09-24 US disclosed
WO-1996000728-A1 PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF CYCLIC UREA HIV PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-01-11 WO disclosed
EP-0686151-A1 SUBSTITUTED CYCLIC CARBONYLS AND DERIVATIVES THEREOF USEFUL AS RETROVIRAL PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-12-13 EP disclosed
US-5466797-A Intermediates for the preparation of cyclic urea THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-11-14 US disclosed
WO-1994019329-A1 SUBSTITUTED CYCLIC CARBONYLS AND DERIVATIVES THEREOF USEFUL AS RETROVIRAL PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1994-09-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070105899-A1 Benzene compounds ACACB, ACACA, FABP4 ALDH1A1 115/4885RECQL 2474/4885NR1I2 473/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.