SCHEMBL4823327

SCHEMBL4823327

NC(=O)c1ccc2cccc(N)c2n1

nearest known ligand 0.69

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 1/20 0.69
KDM4E B2RXH2 1/20 0.47
KMT2A Q03164 1/20 0.47
PARP1 P09874 5/20 0.45
HTR3A P46098 1/20 0.44
PLAU P00749 3/20 0.39
NCF1 P14598 1/20 0.39
MMP2 P08253 2/20 0.39
GRM2 Q14416 1/20 0.36
CCNC P24863 1/20 0.36
CDK8 P49336 1/20 0.36
F2 P00734 1/20 0.36
PLG P00747 1/20 0.36
PLAT P00750 1/20 0.36
KLK1 P06870 1/20 0.36
PRSS1 P07477 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Carbamic Acid SCHEMBL2670938 0.86 KDM4E (0.62) PIM1KDM4EKMT2AMMP2
SCHEMBL3388245 0.85 KDM4E (0.66) PIM1KDM4EKMT2AMMP2
SCHEMBL29831204 0.85 KDM4E (0.66) PIM1KDM4EKMT2AMMP2
SCHEMBL14610232 0.82 PIM1 (0.68) PIM1KDM4EKMT2APARP1GRM2
SCHEMBL2670940 0.82 PIM1 (0.47) PIM1KDM4EKMT2APARP1HTR3A
SCHEMBL3182339 0.81 PIM1 (1.00) PIM1KDM4EKMT2APARP1PLAU
SCHEMBL13977541 0.80 PIM1 (0.67) PIM1KDM4EKMT2APARP1MMP2
SCHEMBL28346452 0.80 PIM1 (0.45) PIM1KDM4EKMT2APARP1HTR3A
SCHEMBL4819927 0.80 ALDH1A1 (0.46) PIM1KDM4EKMT2AMMP2
SCHEMBL27998643 0.80 CNR2 (0.58) PIM1KDM4EKMT2AMMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-121758365-A Preparation method of 5-difluoro alkyl-8-amino quinoline amide compound 阜阳师范大学 2026-03-31 CN disclosed
CN-1659144-B Quinoline and isoquinoline derivatives, process for their preparation and their use as inflammation inhibitors SCHERING AG 2010-09-08 CN disclosed
US-7329753-B2 Quinoline and isoquinoline derivatives, a process for their production and their use as inflammation inhibitors SCHERING AG (DE) 2008-02-12 US disclosed
US-20060229333-A1 Quinoline and isoquinoline derivatives, a process for their production and their use as inflammation inhibitors BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2006-10-12 US disclosed
US-7109212-B2 Quinoline and isoquinoline derivatives, a process for their production and their use as inflammation inhibitors SCHERING AG (DE) 2006-09-19 US disclosed
CN-1659144-A Quinoline and isoquinoline derivatives, process for their preparation and their use as inflammation inhibitors SCHERING AG (DE) 2005-08-24 CN disclosed
US-20050165050-A1 Quinoline and isoquinoline derivatives, a process for their production and their use as inflammation inhibitors BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2005-07-28 US disclosed
US-6897224-B2 Quinoline and isoquinoline derivatives, a process for their production and their use as inflammation inhibitors SCHERING AG (DE) 2005-05-24 US disclosed
US-20040116694-A1 Quinoline and isoquinoline derivatives, a process for their production and their use as inflammation inhibitors SCHERING AG (DE) 2004-06-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060229333-A1 Quinoline and isoquinoline derivatives, a process for their production and their use as inflammation inhibitors NFKBIA, IL1B, IRF3 PIM1 1159/4885KDM4E 3072/4885KMT2A 3773/4885
US-20050165050-A1 Quinoline and isoquinoline derivatives, a process for their production and their use as inflammation inhibitors NFKBIA, IL1B, IRF3 PIM1 1159/4885KDM4E 3072/4885KMT2A 3773/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.