SCHEMBL482356

SCHEMBL482356

COc1ccccc1Nc1ccc([N+](=O)[O-])c(-c2cccc(O)c2)n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.53
MAPK1 P28482 3/20 0.53
MAPT P10636 9/20 0.51
PKM P14618 1/20 0.51
TDP1 Q9NUW8 3/20 0.49
L3MBTL1 Q9Y468 2/20 0.49
LMNA P02545 2/20 0.49
SMN1; SMN2 Q16637 1/20 0.48
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
RAB9A P51151 2/20 0.47
RECQL P46063 2/20 0.47
GAA P10253 2/20 0.45
NPC1 O15118 1/20 0.45
DUSP3 P51452 1/20 0.43
PTPN5 P54829 1/20 0.43
PTPN11 Q06124 1/20 0.43
MAPK10 P53779 1/20 0.43
BRAF P15056 1/20 0.42
EGFR P00533 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2209657 0.82 MEN1 (0.56) ALDH1A1MAPK1MAPTPKMTDP1
SCHEMBL27539926 0.78 MAPK1 (0.64) ALDH1A1MAPK1MAPTPKMTDP1
SCHEMBL481887 0.77 MAPT (0.50) ALDH1A1MAPK1MAPTPKMTDP1
SCHEMBL4940856 0.70 L3MBTL1 (0.68) ALDH1A1MAPK1MAPTPKMTDP1
SCHEMBL30819288 0.70 L3MBTL1 (0.68) ALDH1A1MAPK1MAPTPKMTDP1
SCHEMBL10711270 0.69 L3MBTL1 (0.67) ALDH1A1MAPK1MAPTPKMTDP1
SCHEMBL8938823 0.69 MAPK1 (0.61) ALDH1A1MAPK1MAPTPKMTDP1
SCHEMBL481445 0.69 KMT2A (0.65) ALDH1A1MAPK1MAPTPKMTDP1
SCHEMBL14247580 0.68 MAPK1 (0.60) ALDH1A1MAPK1MAPTPKMTDP1
SCHEMBL14053276 0.67 HSP90AA1 (0.49) ALDH1A1MAPTPKMTDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2078016-B1 HETEROARYL COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH SIGNAL PHARM LLC (US) 2012-02-01 EP disclosed