SCHEMBL4824475

SCHEMBL4824475

C#CCN.O=C(O)c1csc(-c2c(-c3ccc(F)cc3)n[nH]c2C2CCN(C(=O)CO)CC2)n1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPK11 Q15759 15/20 0.51
MAPK14 Q16539 15/20 0.51
KCNH2 Q12809 1/20 0.48
MAP4K4 O95819 1/20 0.40
EGFR P00533 1/20 0.40
PRKACA P17612 1/20 0.40
FRK P42685 1/20 0.40
MAPK9 P45984 1/20 0.40
CSNK1A1 P48729 1/20 0.40
CSNK1D P48730 1/20 0.40
MINK1 Q8N4C8 1/20 0.40
CPT1A P50416 1/20 0.34
IRAK4 Q9NWZ3 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6004425 0.94 MAPK11 (0.56) MAPK11MAPK14KCNH2MAP4K4EGFR
SCHEMBL6002821 0.88 MAPK11 (0.49) MAPK11MAPK14KCNH2MAP4K4EGFR
SCHEMBL4824481 0.86 MAPK11 (0.47) MAPK11MAPK14KCNH2MAP4K4EGFR
SCHEMBL6004539 0.83 MAPK11 (0.51) MAPK11MAPK14KCNH2MAP4K4EGFR
SCHEMBL4761930 0.83 MAPK11 (0.51) MAPK11MAPK14KCNH2MAP4K4EGFR
SCHEMBL4761929 0.82 MAPK11 (0.50) MAPK11MAPK14KCNH2MAP4K4EGFR
SCHEMBL4761505 0.80 MAPK11 (0.52) MAPK11MAPK14KCNH2
SCHEMBL3373577 0.80 MAPK11 (0.59) MAPK11MAPK14KCNH2MAPK9
Isopropylamine SCHEMBL4827262 0.78 MAPK11 (0.49) MAPK11MAPK14KCNH2
SCHEMBL6004578 0.78 MAPK11 (0.54) MAPK11MAPK14KCNH2CSNK1DIRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1871770-A1 ORTHO-TERPHENYL INHIBITORS OF P38 KINASE AND METHODS OF TREATING INFLAMMATORY DISORDERS Kalypsys, Inc. (US) 2008-01-02 EP disclosed
WO-2006116355-A1 ORTHO-TERPHENYL INHIBITORS OF P38 KINASE AND METHODS OF TREATING INFLAMMATORY DISORDERS KALYPSYS, INC. (US) 2006-11-02 WO disclosed