SCHEMBL4824898

SCHEMBL4824898

O=C(N[C@@H](Cc1ccc(-c2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1)C(=O)O)c1cc2ccccc2cc1O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIFC1 Q9BW19 5/20 0.57
CDK2 P24941 1/20 0.51
GPR34 Q9UPC5 1/20 0.51
MME P08473 3/20 0.47
ACE P12821 3/20 0.47
ACE2 Q9BYF1 3/20 0.47
CPA1 P15085 2/20 0.47
ITGB1 P05556 1/20 0.46
ITGA4 P13612 1/20 0.46
FPR2 P25090 1/20 0.45
RXRA P19793 1/20 0.44
RXRB P28702 1/20 0.44
RXRG P48443 1/20 0.44
HPGDS O60760 1/20 0.44
PIN1 Q13526 1/20 0.44
PDK1 Q15118 1/20 0.44
PDK2 Q15119 1/20 0.44
PDK3 Q15120 1/20 0.44
PDK4 Q16654 1/20 0.44
MCL1 Q07820 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4833896 0.94 KIFC1 (0.56) KIFC1CDK2GPR34MMEACE
SCHEMBL4833892 0.94 KIFC1 (0.56) KIFC1CDK2GPR34MMEACE
SCHEMBL27611059 0.89 MME (0.57) MMEACEACE2CPA1ITGB1
SCHEMBL5926558 0.89 MME (0.57) MMEACEACE2CPA1ITGB1
SCHEMBL6406839 0.89 KDR (0.54) KIFC1CDK2GPR34
SCHEMBL4831843 0.87 FPR2 (0.56) KIFC1GPR34MMEACEACE2
SCHEMBL4831835 0.87 FPR2 (0.56) KIFC1GPR34MMEACEACE2
SCHEMBL5927070 0.84 KIFC1 (0.61) KIFC1GPR34MMEACEACE2
SCHEMBL6098431 0.83 KIFC1 (0.69) KIFC1CDK2GPR34MMEITGB1
SCHEMBL5927352 0.83 KIFC1 (0.61) KIFC1CDK2GPR34MMEACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7459472-B2 Aryl and heteroaryl compounds, compositions, and methods of use TRANSTECH PHARMA, INC. (US) 2008-12-02 US disclosed