SCHEMBL4826506

SCHEMBL4826506

NCCC(C(N)=O)c1ccc(Cl)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABBR2 O75899 6/20 0.46
GABBR1 Q9UBS5 6/20 0.46
CYP2C9 P11712 3/20 0.46
LMNA P02545 3/20 0.46
KMT2A Q03164 3/20 0.46
CYP2D6 P10635 2/20 0.46
CYP2C19 P33261 2/20 0.46
MEN1 O00255 2/20 0.46
CYP1A2 P05177 2/20 0.46
THRB P10828 2/20 0.46
CYP3A4 P08684 1/20 0.46
ADORA3 P0DMS8 1/20 0.46
NFKB1 P19838 1/20 0.46
DRD3 P35462 1/20 0.46
BLM P54132 1/20 0.46
TSHR P16473 1/20 0.46
SLC6A4 P31645 1/20 0.42
SLC6A3 Q01959 1/20 0.42
MAPT P10636 1/20 0.41
PMP22 Q01453 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4830664 0.85 CYP2C9 (0.51) GABBR2GABBR1CYP2C9LMNAKMT2A
SCHEMBL10255978 0.85 GABBR2 (0.53) GABBR2GABBR1CYP2C9LMNAKMT2A
SCHEMBL3637896 0.84 FFAR2 (0.50) GABBR2GABBR1CYP2C9LMNAKMT2A
SCHEMBL11082974 0.84 CYP2C9 (0.42) GABBR2GABBR1CYP2C9LMNAKMT2A
Hydrochloric Acid SCHEMBL22831450 0.84 CYP2C9 (0.50) GABBR2GABBR1CYP2C9LMNAKMT2A
SCHEMBL9328610 0.83 ESR1 (0.44) CYP2C9LMNAKMT2ACYP2D6CYP2C19
SCHEMBL28419253 0.82 CYP2C9 (0.49) GABBR2GABBR1CYP2C9LMNAKMT2A
Hydrochloric Acid SCHEMBL326728 0.81 TDP1 (0.46) CYP2C9LMNAKMT2ACYP2D6CYP2C19
SCHEMBL13357525 0.81 CDC7 (0.49) LMNACYP2D6CYP3A4SLC6A4SLC6A3
SCHEMBL3642653 0.80 FFAR2 (0.50) GABBR2GABBR1CYP2C9LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7402652-B2 Baclofen conjugate and a pharmaceutical composition for treatment of neuronal disorders MILLER LANDON C G 2008-07-22 US disclosed
US-20060058221-A1 Baclofen conjugate and a pharmaceutical composition for treatment of neuronal disorders MILLER LANDON C 2006-03-16 US disclosed