SCHEMBL9328610

SCHEMBL9328610

NCCC(C(N)=O)c1ccc(O)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.44
ESR2 Q92731 4/20 0.44
TAAR1 Q96RJ0 4/20 0.44
HTR3A P46098 2/20 0.44
HIF1A Q16665 2/20 0.44
TSHR P16473 1/20 0.44
NFKB1 P19838 1/20 0.44
TDP1 Q9NUW8 4/20 0.42
KDM4E B2RXH2 3/20 0.42
ALOX15 P16050 2/20 0.42
APEX1 P27695 1/20 0.42
EPHX1 P07099 1/20 0.42
GRM8 O00222 1/20 0.40
GRM4 Q14833 1/20 0.40
CA2 P00918 1/20 0.39
LMNA P02545 2/20 0.38
SLC6A2 P23975 2/20 0.38
CYP2C19 P33261 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HTR1A P08908 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL326728 0.98 TDP1 (0.46) ESR1ESR2TAAR1HTR3AHIF1A
SCHEMBL15653352 0.86 ESR1 (0.46) ESR1ESR2TAAR1HTR3AHIF1A
SCHEMBL21357582 0.85 ESR1 (0.44) ESR1ESR2TAAR1HTR3AHIF1A
SCHEMBL3253687 0.84 TAAR1 (0.52) ESR1ESR2TAAR1HTR3AHIF1A
SCHEMBL4826506 0.83 GABBR2 (0.46) TSHRNFKB1EPHX1LMNACYP2C19
SCHEMBL4938891 0.83 ESR1 (0.47) ESR1ESR2TAAR1HTR3AHIF1A
SCHEMBL27691659 0.82 EPHX1 (0.61) TAAR1EPHX1LMNACYP2C19CYP1A2
SCHEMBL3466433 0.80 ESR1 (0.47) ESR1ESR2TAAR1HTR3AHIF1A
SCHEMBL30368876 0.79 ESR1 (0.40) ESR1ESR2TAAR1HTR3AHIF1A
SCHEMBL4943215 0.78 LMNA (0.54) ESR1ESR2TAAR1HTR3AHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5356894-A Adenosine antagonists SYNGENTA LIMITED (GB) 1994-10-18 US disclosed
US-5270311-A [1,2,4]-Triazolo[1,5-a]and pyrazolo[2,3-a][1,3,5]triazine derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-12-14 US disclosed
CN-1056879-A Pyrrole derivative and preparation method thereof ICI PLC (GB) 1991-12-11 CN disclosed
EP-0459702-A1 Azole Derivatives ZENECA LIMITED (GB) 1991-12-04 EP disclosed