SCHEMBL4827255

SCHEMBL4827255

Cc1cnn(Cc2ccc(C(=O)Nc3cc(F)ccc3Nc3ccccc3)cc2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.55
POLB P06746 1/20 0.55
RAB9A P51151 4/20 0.52
SMN1; SMN2 Q16637 4/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
HTT P42858 3/20 0.52
GAA P10253 2/20 0.52
LMNA P02545 6/20 0.49
NAMPT P43490 1/20 0.49
MAPT P10636 4/20 0.49
KMT2A Q03164 4/20 0.48
MEN1 O00255 3/20 0.48
MAPK1 P28482 1/20 0.48
TAS2R8 Q9NYW2 1/20 0.45
KDM4E B2RXH2 1/20 0.45
HDAC3 O15379 1/20 0.44
JAK2 O60674 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3558592 0.83 ALDH1A1 (0.59) ALDH1A1POLBRAB9ASMN1; SMN2L3MBTL1
SCHEMBL3555192 0.77 ALDH1A1 (0.61) ALDH1A1POLBRAB9ASMN1; SMN2L3MBTL1
SCHEMBL3554578 0.71 HDAC1 (0.47) ALDH1A1POLBSMN1; SMN2LMNAMAPT
SCHEMBL19087149 0.70 HSD17B10 (0.70) ALDH1A1POLBSMN1; SMN2L3MBTL1GAA
SCHEMBL3553873 0.69 HDAC1 (0.63) ALDH1A1RAB9ASMN1; SMN2L3MBTL1HTT
SCHEMBL3556580 0.68 HDAC1 (0.62) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL3549681 0.68 HDAC2 (0.59) ALDH1A1POLBSMN1; SMN2LMNAMAPT
SCHEMBL130830 0.67 L3MBTL1 (0.62) ALDH1A1POLBRAB9ASMN1; SMN2L3MBTL1
SCHEMBL17221323 0.67 KLKB1 (0.56) ALDH1A1RAB9AL3MBTL1GAALMNA
SCHEMBL4516147 0.67 LMNA (0.70) ALDH1A1POLBRAB9ASMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904452-A2 HISTONE DEACETYLASE INHIBITORS Takeda San Diego, Inc. (US) 2008-04-02 EP claimed
WO-2007011626-A2 HISTONE DEACETYLASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2007-01-25 WO claimed