SCHEMBL4829931

SCHEMBL4829931

O=C(Nc1ccc(S(=O)(=O)N[C@H](C(=O)O)c2ccccc2)cc1)c1ccccc1

nearest known ligand 0.67

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MMP9 P14780 4/20 0.67
MMP2 P08253 1/20 0.67
PRMT1 Q99873 2/20 0.60
MEN1 O00255 2/20 0.59
KMT2A Q03164 2/20 0.59
HDAC8 Q9BY41 1/20 0.58
HDAC6 Q9UBN7 1/20 0.58
LMNA P02545 1/20 0.58
CA1 P00915 2/20 0.57
CA2 P00918 2/20 0.57
CA12 O43570 1/20 0.57
CA9 Q16790 1/20 0.57
HPGD P15428 1/20 0.57
HPN P05981 2/20 0.55
PLAU P00749 1/20 0.55
POLB P06746 1/20 0.53
ALDH1A1 P00352 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4824739 0.91 MEN1 (0.58) MMP9MMP2MEN1KMT2AHPGD
SCHEMBL4826124 0.91 MMP9 (0.71) MMP9MMP2MEN1KMT2ALMNA
SCHEMBL4833932 0.88 LMNA (0.69) MMP9MMP2MEN1KMT2ALMNA
SCHEMBL4832393 0.88 MMP9 (0.68) MMP9MMP2MEN1KMT2ALMNA
SCHEMBL2053891 0.82 SLC1A3 (0.56) MMP9MMP2MEN1KMT2AHDAC8
SCHEMBL10102615 0.82 SLC1A3 (0.56) MMP9MMP2MEN1KMT2AHDAC8
SCHEMBL7663210 0.82 MMP9 (0.76) MMP9MMP2PRMT1MEN1KMT2A
SCHEMBL7669616 0.82 MMP9 (0.76) MMP9MMP2PRMT1MEN1KMT2A
SCHEMBL7668862 0.81 MMP9 (1.00) MMP9MMP2POLBALDH1A1
SCHEMBL7675244 0.81 MMP9 (1.00) MMP9MMP2POLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6403644-B1 FOR PREVENTION AND/OR TREATMENT OF DISEASES INDUCED BY OVEREXPRESSION AND EXCESS ACTIVITY OF MATRIX METALLOPROTEINASE; FOR EXAMPLE, RHEUMATOID, ARTHROSTEITIS, UNUSUAL BONE RESORPTION, OSTEOPOROSIS, PERIODONTITIS ONO PHARMACEUTICAL CO., LTD. (JP) 2002-06-11 US claimed
EP-0757037-A2 Sulfonylamino acid derivatives as metalloproteinase inhibitors ONO PHARMACEUTICAL CO., LTD. (JP) 1997-02-05 EP claimed
US-7335686-B2 Method and composition for treating osteoporosis COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2008-02-26 US disclosed
EP-1678124-A1 NOVEL MOLECULES TO DEVELOP DRUG FOR THE TREATMENT OF OSTEOPOROSIS COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2006-07-12 EP disclosed
WO-2005037774-A1 NOVEL MOLECULES TO DEVELOP DRUG FOR THE TREATMENT OF OSTEOPOROSIS COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2005-04-28 WO disclosed
US-20050085537-A1 Method and composition for treating osteoporosis COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2005-04-21 US disclosed
US-6403644-B1 FOR PREVENTION AND/OR TREATMENT OF DISEASES INDUCED BY OVEREXPRESSION AND EXCESS ACTIVITY OF MATRIX METALLOPROTEINASE; FOR EXAMPLE, RHEUMATOID, ARTHROSTEITIS, UNUSUAL BONE RESORPTION, OSTEOPOROSIS, PERIODONTITIS ONO PHARMACEUTICAL CO., LTD. (JP) 2002-06-11 US disclosed
US-6177466-B1 Sulfonylamino acid derivatives ONO PHARMACEUTICAL CO., LTD. (JP) 2001-01-23 US disclosed
EP-0757037-A2 Sulfonylamino acid derivatives as metalloproteinase inhibitors ONO PHARMACEUTICAL CO., LTD. (JP) 1997-02-05 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050085537-A1 Method and composition for treating osteoporosis SOST, CALCR, MSR1 MMP9 2131/4885MMP2 2736/4885PRMT1 733/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.