SCHEMBL4831359

SCHEMBL4831359

CN(CC1Cc2cc(F)cc(-c3cccnc3)c2O1)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AQP1 P29972 3/20 0.39
GBA1 P04062 7/20 0.38
KDM4E B2RXH2 1/20 0.38
USP2 O75604 1/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
TSHR P16473 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CYP11B1 P15538 3/20 0.37
CYP11B2 P19099 3/20 0.37
MAOA P21397 1/20 0.35
GPR84 Q9NQS5 1/20 0.33
PDE4B Q07343 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4968896 0.81 AQP1 (0.43) AQP1
SCHEMBL4224624 0.81 AQP1 (0.55) AQP1CYP11B1CYP11B2MAOAPDE4B
SCHEMBL4230606 0.80 AQP1 (0.61) AQP1CYP11B1CYP11B2MAOAPDE4B
SCHEMBL4837073 0.80 AQP1 (0.44) AQP1
SCHEMBL4230613 0.79 AQP1 (0.45) AQP1CYP11B1CYP11B2MAOAPDE4B
SCHEMBL4830417 0.78 AQP1 (0.65) AQP1
SCHEMBL4965176 0.78 AQP1 (0.41) AQP1
SCHEMBL4597059 0.77 PARP1 (0.47) AQP1CYP11B1CYP11B2MAOAGPR84
SCHEMBL4788915 0.77 AQP1 (0.53) AQP1KDM4EUSP2
SCHEMBL4597056 0.75 TDO2 (0.38) AQP1CYP11B1CYP11B2MAOAGPR84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1871355-A1 NEW THERAPEUTIC COMBIANATIONS FOR THE TREATMENT OR PREVENTION OF DEPRESSION Wyeth (US) 2008-01-02 EP disclosed
WO-2006116149-A1 NEW THERAPEUTIC COMBIANATIONS FOR THE TREATMENT OR PREVENTION OF DEPRESSION WYETH (US) 2006-11-02 WO disclosed