SCHEMBL4833706

SCHEMBL4833706

Nc1ccc(Cn2ncnn2)cc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.41
CYP11B2 P19099 2/20 0.41
ALDH1A1 P00352 2/20 0.40
HTR1A P08908 1/20 0.40
HTR2C P28335 1/20 0.40
HDAC6 Q9UBN7 1/20 0.38
CYP3A4 P08684 2/20 0.38
GFER P55789 1/20 0.38
TSHR P16473 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
LMNA P02545 1/20 0.38
LOXL2 Q9Y4K0 1/20 0.37
CYP19A1 P11511 3/20 0.36
CYP17A1 P05093 1/20 0.36
HTR6 P50406 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
ADORA2A P29274 1/20 0.35
S1PR1 P21453 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9697609 0.98 CYP11B1 (0.40) CYP11B1CYP11B2ALDH1A1HTR1AHTR2C
SCHEMBL8784962 0.80 CYP19A1 (0.57) CYP11B1CYP11B2HTR1AHTR2CCYP19A1
SCHEMBL10288500 0.79 CYP19A1 (0.47) CYP11B1CYP11B2ALDH1A1TSHRCYP19A1
SCHEMBL932804 0.77 HTR1A (0.37) HTR1AHTR2CCYP19A1HRH3S1PR1
SCHEMBL31272207 0.77 POLB (0.40) ALDH1A1HTR1AHTR2CTSHRLMNA
SCHEMBL15542865 0.77 ALDH1A1 (0.47) CYP11B1CYP11B2ALDH1A1GFERLMNA
SCHEMBL2351887 0.77 CYP19A1 (0.64) CYP11B1CYP11B2LOXL2CYP19A1
SCHEMBL3142438 0.75 CYP19A1 (0.61) CYP11B1CYP11B2ALDH1A1HDAC6CYP3A4
SCHEMBL4834371 0.74 CYP19A1 (0.48) ALDH1A1TSHRTDP1LMNALOXL2
SCHEMBL15542806 0.68 CYP11B1 (0.46) CYP11B1CYP11B2ALDH1A1HTR1AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080287438-A1 Agent for preventing or treating neuropathy MOMOSE YU 2008-11-20 US disclosed
US-7423159-B2 Agent for preventing or treating neuropathy TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-09 US disclosed
CN-1731994-A Prophylactic and therapeutic agent for neuropathy TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2006-02-08 CN disclosed
US-20060004069-A1 Agent for preventing or treating neuropathy TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2006-01-05 US disclosed
EP-1556032-A1 AGENT FOR PREVENTING OR TREATING NEUROPATHY Takeda Pharmaceutical Company Limited (JP) 2005-07-27 EP disclosed
WO-2004039365-A1 AGENT FOR PREVENTING OR TREATING NEUROPATHY TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2004-05-13 WO disclosed
EP-0497512-B1 Imidazole, triazole and tetrazole derivatives MERCK SHARP & DOHME (GB) 1997-09-24 EP disclosed
EP-0778275-A1 Process for the preparation of imidazole, triazole and tetrazole derivatives and their use as selective 5-HT-1 receptor agonists MERCK SHARP & DOHME LTD. (GB) 1997-06-11 EP disclosed
US-5602162-A TREATMENT AND/OR PREVENTION OF MIGRAINE MERCK, SHARP & DOHME LTD. (GB) 1997-02-11 US disclosed
US-5451588-A Treatment of migraines MERCK SHARP & DOHME LTD. (GB) 1995-09-19 US disclosed
US-5298520-A Triazole containing indole derivatives MERCK SHARP & DOHME LIMITED (GB) 1994-03-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060004069-A1 Agent for preventing or treating neuropathy NR2C2, NR0B2, NR2E1 CYP11B1 377/4885CYP11B2 90/4885ALDH1A1 2652/4885
US-20080287438-A1 Agent for preventing or treating neuropathy NR2C2, NR0B2, NR2E1 CYP11B1 377/4885CYP11B2 90/4885ALDH1A1 2652/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.