SCHEMBL484005

SCHEMBL484005

O=C=Nc1ccccc1N=C=S

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 0.52
ALDH1A1 P00352 4/20 0.52
HPGD P15428 3/20 0.52
TDP1 Q9NUW8 3/20 0.52
ABCB11 O95342 1/20 0.52
NR3C1 P04150 1/20 0.52
CYP1A2 P05177 1/20 0.52
ADRA2A P08913 1/20 0.52
ADORA3 P0DMS8 1/20 0.52
ALOX15 P16050 1/20 0.52
ADRA2C P18825 1/20 0.52
MAOA P21397 1/20 0.52
DRD1 P21728 1/20 0.52
SLC6A4 P31645 1/20 0.52
HTR2B P41595 1/20 0.52
CCR2 P41597 1/20 0.52
HSD17B10 Q99714 1/20 0.52
POLB P06746 1/20 0.47
MIF P14174 5/20 0.46
APLNR P35414 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29374052 0.87 ALDH1A1 (0.62) CYP3A4ALDH1A1HPGDTDP1ABCB11
SCHEMBL207554 0.87 ALDH1A1 (0.62) CYP3A4ALDH1A1HPGDTDP1ABCB11
SCHEMBL15431 0.87 CYP3A4 (0.64) CYP3A4ALDH1A1HPGDTDP1ABCB11
SCHEMBL29395383 0.87 CYP3A4 (0.64) CYP3A4ALDH1A1HPGDTDP1ABCB11
Benzene SCHEMBL28766229 0.85 CYP3A4 (0.61) CYP3A4ALDH1A1HPGDTDP1ABCB11
SCHEMBL30244709 0.85 CYP3A4 (0.61) CYP3A4ALDH1A1HPGDTDP1ABCB11
Ammonia Solution, Strong SCHEMBL28158244 0.85 CYP3A4 (0.61) CYP3A4ALDH1A1HPGDTDP1ABCB11
Fluoride SCHEMBL28813057 0.85 CYP3A4 (0.61) CYP3A4ALDH1A1HPGDTDP1ABCB11
Water SCHEMBL28526910 0.85 CYP3A4 (0.61) CYP3A4ALDH1A1HPGDTDP1ABCB11
SCHEMBL28944561 0.84 CYP3A4 (0.40) CYP3A4ALDH1A1HPGDTDP1ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411433-A1 POLYURETHANES, ARTICLES AND COATINGS PREPARED THEREFROM AND METHODS OF MAKING THE SAME PPG Industries Ohio, Inc. (US) 2012-02-01 EP disclosed
WO-2010110784-A1 POLYURETHANES, ARTICLES AND COATINGS PREPARED THEREFROM AND METHODS OF MAKING THE SAME PPG INDUSTRIES OHIO, INC. (US) 2010-09-30 WO disclosed
US-7144989-B2 Pegylated non-hypertensive hemoglobins, methods of preparing same, and uses thereof ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2006-12-05 US disclosed
US-7084112-B2 Activated polyethylene glycol compounds ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2006-08-01 US disclosed
US-6962954-B2 Activated polyethylene glycol compounds ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2005-11-08 US disclosed
US-20050159339-A1 Pegylated non-hypertensive hemoglobins, methods of preparing same, and uses thereof ALBERT EINSTEIN COLLEGE OF MEDICINE, INC. 2005-07-21 US disclosed
US-20040147736-A1 Activated polyethylene glycol compounds ALBERT EINSTEIN COLLEGE OF MEDICINE, INC. 2004-07-29 US disclosed
US-20040127697-A1 Activated polyethylene glycol compounds ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY 2004-07-01 US disclosed
US-6737524-B2 ARYL ISOTHIOCYANATE DERIVATIVES; ATTACHING TO BIOMOLECULES SUCH AS PROTEINS OR PEPTIDES; ENHANCING IN VIVO CIRCULATION HALFLIFE Smith, Paul K. 2004-05-18 US disclosed
US-20030187248-A1 Activated polyethylene glycol compounds ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY 2003-10-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030187248-A1 Activated polyethylene glycol compounds ADH1C, PIGO, AADAC CYP3A4 1790/4885ALDH1A1 547/4885HPGD 2705/4885
US-20040127697-A1 Activated polyethylene glycol compounds ADH1C, PIGO, AADAC CYP3A4 1790/4885ALDH1A1 547/4885HPGD 2705/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.