SCHEMBL4840147

SCHEMBL4840147

COc1ccc(N(C(=O)Nc2cccc(F)c2)c2ccnc(N[C@@H](C)C(C)(C)O)n2)cc1

nearest known ligand 0.70

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 12/20 0.70
SMN1; SMN2 Q16637 2/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
POLB P06746 1/20 0.42
KMT2A Q03164 1/20 0.42
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
KDR P35968 2/20 0.39
PDGFRA P16234 1/20 0.39
LCK P06239 1/20 0.38
SRC P12931 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4840138 1.00 MAPK14 (0.70) MAPK14SMN1; SMN2NPC1RAB9APOLB
SCHEMBL4840708 0.92 MAPK14 (0.72) MAPK14SMN1; SMN2NPC1RAB9APOLB
SCHEMBL4840721 0.92 MAPK14 (0.72) MAPK14SMN1; SMN2NPC1RAB9APOLB
SCHEMBL4840534 0.91 MAPK14 (0.73) MAPK14SMN1; SMN2NPC1RAB9ATP53
SCHEMBL4840530 0.91 MAPK14 (0.73) MAPK14SMN1; SMN2NPC1RAB9ATP53
SCHEMBL4838892 0.91 MAPK14 (0.67) MAPK14SMN1; SMN2NPC1RAB9APOLB
SCHEMBL4838900 0.91 MAPK14 (0.67) MAPK14SMN1; SMN2NPC1RAB9APOLB
SCHEMBL4836187 0.90 MAPK14 (0.73) MAPK14SMN1; SMN2NPC1RAB9APOLB
SCHEMBL4836181 0.90 MAPK14 (0.73) MAPK14SMN1; SMN2NPC1RAB9APOLB
SCHEMBL4828771 0.90 MAPK14 (0.71) MAPK14KDRLCKSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7402589-B2 Tri-substituted ureas as cytokine inhibitors THE PROCTER & GAMBLE COMPANY (US) 2008-07-22 US claimed
US-20050245555-A1 Tri-substituted ureas as cytokine inhibitors THE PROCTER & GAMBLE COMPANY (US) 2005-11-03 US claimed
US-7402589-B2 Tri-substituted ureas as cytokine inhibitors THE PROCTER & GAMBLE COMPANY (US) 2008-07-22 US disclosed
US-20050245555-A1 Tri-substituted ureas as cytokine inhibitors THE PROCTER & GAMBLE COMPANY (US) 2005-11-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050245555-A1 Tri-substituted ureas as cytokine inhibitors IL1B, IL1A, IL6 MAPK14 2674/4885SMN1; SMN2 4628/4885NPC1 3402/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.