SCHEMBL4841972

SCHEMBL4841972

C[Si](C)(C)CCOCn1c(N2CCNCC2)nc(-c2ccc(C(F)(F)F)cc2)c1-c1ccc(C(F)(F)F)cc1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 5/20 0.44
PRMT5 O14744 1/20 0.36
KCNH2 Q12809 3/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
DGAT1 O75907 1/20 0.35
KDM1A O60341 2/20 0.35
DRD2 P14416 1/20 0.35
HTR6 P50406 1/20 0.35
PIM1 P11309 1/20 0.34
PIM3 Q86V86 1/20 0.34
PIM2 Q9P1W9 1/20 0.34
HTR3A P46098 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4841841 0.92 SOS1 (0.42) SOS1PRMT5KCNH2HTR2CKDM1A
SCHEMBL5201999 0.82 EPHX2 (0.44)
SCHEMBL4843896 0.81 TRPV1 (0.44)
SCHEMBL4853070 0.80 HTR2C (0.38) SOS1HTR2CKDM1AHTR3A
SCHEMBL4842017 0.75 TRPV1 (0.40)
SCHEMBL5185302 0.75 TRPV1 (0.40)
SCHEMBL5201005 0.74 HTR2C (0.34) SOS1HTR2CKDM1APIM1
SCHEMBL4842921 0.71 HTR2C (0.38) SOS1HTR2CKDM1APIM1
SCHEMBL4849012 0.71 TRPV1 (0.44)
SCHEMBL4847436 0.69 HTR2C (0.36) SOS1HTR2CPIM1HTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7439360-B2 Vanilloid receptor ligands and their use in treatments AMGEN INC. (US) 2008-10-21 US disclosed
US-7439360-B2 Vanilloid receptor ligands and their use in treatments AMGEN INC. (US) 2008-10-21 US disclosed
US-20060084640-A1 Vanilloid receptor ligands and their use in treatments AMGEN INC. 2006-04-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060084640-A1 Vanilloid receptor ligands and their use in treatments TRPV1, TRPV3, TRPV2 SOS1 2211/4885PRMT5 4414/4885KCNH2 299/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.