SCHEMBL4828449

SCHEMBL4828449

O=C(Oc1nn(C(=O)N2CCC(C(F)(F)F)CC2)c2cc(F)ccc12)ON1CCC(C(F)(F)F)CC1

nearest known ligand 0.39

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SPR P35270 7/20 0.34
RBP4 P02753 4/20 0.34
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2956860 0.88 SPR (0.36) SPRRBP4
SCHEMBL16242496 0.86 SPR (0.32) SPRHPGD
SCHEMBL4837047 0.82 NPC1 (0.36)
SCHEMBL16242493 0.79 FAAH (0.42)
SCHEMBL4829941 0.76 GRM4 (0.34) HPGD
SCHEMBL2955527 0.76 GAA (0.43) RBP4HPGD
SCHEMBL2966049 0.74 GAA (0.38) SPRHPGD
SCHEMBL16242373 0.73 HPGD (0.34) HPGD
SCHEMBL1573644 0.73 RAB9A (0.39) RBP4HPGD
SCHEMBL2965248 0.71 NPC1 (0.36) HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937648-B1 DIACYL INDAZOL DERIVATIVES AS LIPASE AND PHOSPHOLIPASE INHIBITORS SANOFI SA (FR) 2014-11-26 EP disclosed
EP-1937648-A1 DIACYL INDAZOL DERIVATIVES AS LIPASE AND PHOSPHOLIPASE INHIBITORS sanofi-aventis (FR) 2008-07-02 EP disclosed
WO-2007042178-A1 DIACYL INDAZOL DERIVATIVES AS LIPASE AND PHOSPHOLIPASE INHIBITORS SANOFI-AVENTIS (DE) 2007-04-19 WO disclosed