SCHEMBL4845045

SCHEMBL4845045

CC1Cc2onc(-c3ccccc3O)c2C(=O)C1C(=O)O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.36
RAB9A P51151 5/20 0.36
SMN1; SMN2 Q16637 5/20 0.36
TP53 P04637 3/20 0.36
HPGD P15428 2/20 0.36
NFKB1 P19838 2/20 0.36
NFKB2 Q00653 2/20 0.36
RELA Q04206 2/20 0.36
ALDH1A1 P00352 1/20 0.36
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
HSP90AB1 P08238 1/20 0.36
MAPT P10636 3/20 0.34
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
ACHE P22303 1/20 0.33
DNMT3B Q9UBC3 1/20 0.32
HSP90AA1 P07900 1/20 0.32
PAX8 Q06710 1/20 0.32
AOC1 P19801 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4917582 0.85 MAOA (0.39) RAB9ATP53HPGDALDH1A1MAPT
SCHEMBL14014136 0.68 BRD4 (0.48) NPC1RAB9ASMN1; SMN2TP53HPGD
SCHEMBL13837599 0.63 HSD17B10 (0.54) NPC1SMN1; SMN2HPGDALDH1A1HSP90AB1
SCHEMBL5820169 0.62 EDNRB (0.45) ALDH1A1MEN1KMT2ACYP1A2CYP2C9
SCHEMBL27927955 0.61 HSD17B10 (0.55) ALDH1A1MAPTMEN1KMT2ACYP2C19
SCHEMBL5952009 0.60 ACHE (0.62) SMN1; SMN2HPGDALDH1A1MAPTACHE
SCHEMBL14261867 0.59 ESR1 (0.72) NPC1RAB9ASMN1; SMN2HPGDNFKB1
SCHEMBL5730461 0.58 ESR1 (0.53) NPC1RAB9ASMN1; SMN2TP53HPGD
SCHEMBL5952103 0.58 ACHE (0.59) ALDH1A1MAPTMEN1KMT2AACHE
SCHEMBL13115609 0.57 ACHE (0.68) SMN1; SMN2HPGDALDH1A1MAPTACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1484325-B1 ISOXAZOLE DERIVATIVES AND PROCESS FOR PRODUCING THE SAME JAPAN SCIENCE & TECH AGENCY (JP) 2014-06-18 EP disclosed
US-7453001-B2 Such as, ethyl 3-(2-hydroxyphenyl)-6-methyl4-oxo4,5,6,7-tetrahydrobenzo[d]isoxazole-5-carboxylate; intermediates JAPAN SCIENCE AND TECHNOLOGY AGENCY (JP) 2008-11-18 US disclosed
US-7342036-B2 Isoxazole derivatives and process for producing the same JAPAN SCIENCE AND TECHNOLOGY AGENCY (JP) 2008-03-11 US disclosed
EP-1484325-A1 ISOXAZOLE DERIVATIVES AND PROCESS FOR PRODUCING THE SAME Japan Science and Technology Agency (JP) 2004-12-08 EP disclosed