SCHEMBL4845542

SCHEMBL4845542

COC(CNC(=O)Cc1ccccc1N)OC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.44
HPGD P15428 3/20 0.44
KDM4E B2RXH2 2/20 0.44
RCE1 Q9Y256 1/20 0.44
HCRTR2 O43614 1/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
TAAR1 Q96RJ0 1/20 0.41
LMNA P02545 1/20 0.41
NPSR1 Q6W5P4 1/20 0.40
HTT P42858 1/20 0.40
POLB P06746 1/20 0.39
CFTR P13569 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CCR3 P51677 1/20 0.39
ADRB2 P07550 1/20 0.39
ADRB1 P08588 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5767226 0.82 MEN1 (0.43) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL29097833 0.82 TAAR1 (0.60) ALDH1A1HPGDMEN1KMT2ANPC1
SCHEMBL10700966 0.78 NPC1 (0.55) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL4850673 0.78 CYP2C19 (0.63) ALDH1A1KDM4EMEN1KMT2ANPC1
SCHEMBL2310135 0.76 MEN1 (0.49) ALDH1A1HPGDMEN1KMT2ANPC1
SCHEMBL27973340 0.76 KMT2A (0.52) ALDH1A1HPGDMEN1KMT2ANPC1
SCHEMBL17462497 0.75 MEN1 (0.48) ALDH1A1HPGDMEN1KMT2ANPC1
SCHEMBL22316651 0.74 ALDH1A1 (0.45) ALDH1A1HPGDKDM4ERCE1HCRTR2
SCHEMBL644296 0.74 ALDH1A1 (0.49) ALDH1A1HPGDKDM4ERCE1MEN1
SCHEMBL14278969 0.73 TAAR1 (0.42) ALDH1A1HPGDKDM4ERCE1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7323458-B1 Dihydrobenzodiazepins and their use for treating dyslipidemia MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2008-01-29 US disclosed
EP-1189890-A1 DIHYDROBENZODIAZEPINS AND THEIR USE FOR TREATING DYSLIPIDEMIA MERCK PATENT GmbH (DE) 2002-03-27 EP disclosed
WO-2001002373-A1 DIHYDROBENZODIAZEPINS AND THEIR USE FOR TREATING DYSLIPIDEMIA MERCK PATENT GMBH (DE) 2001-01-11 WO disclosed