SCHEMBL4847962

SCHEMBL4847962

N=C(N)CCc1ccc(F)c(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNMT P11086 1/20 0.43
TAAR1 Q96RJ0 1/20 0.43
DAO P14920 1/20 0.40
IDO1 P14902 6/20 0.40
PIK3CA P42336 1/20 0.40
HTR3E A5X5Y0 1/20 0.39
HTR3B O95264 1/20 0.39
HTR3A P46098 1/20 0.39
HTR3D Q70Z44 1/20 0.39
HTR3C Q8WXA8 1/20 0.39
ITGB3 P05106 1/20 0.38
ITGAV P06756 1/20 0.38
F9 P00740 1/20 0.37
F10 P00742 1/20 0.37
BACE1 P56817 1/20 0.37
MEN1 O00255 1/20 0.37
PLA2G1B P04054 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4718123 0.98 PNMT (0.42) PNMTTAAR1DAOIDO1PIK3CA
SCHEMBL4837866 0.84 DAO (0.39) TAAR1DAOIDO1F10MAPT
SCHEMBL15517814 0.83 PIK3CA (0.47) PNMTTAAR1DAOIDO1PIK3CA
Hydrochloric Acid SCHEMBL4713635 0.82 DAO (0.38) DAOIDO1F10GAAMAPT
SCHEMBL9104006 0.79 CYP2D6 (0.40) IDO1HTR3EHTR3BHTR3AHTR3D
SCHEMBL28107153 0.79 PIK3CA (0.49) PNMTTAAR1DAOPIK3CAMAPT
Hydrochloric Acid SCHEMBL1623226 0.79 IDO1 (0.37) PNMTTAAR1DAOIDO1PIK3CA
Hydrochloric Acid SCHEMBL9107781 0.78 CYP2D6 (0.39) IDO1F10GAAMAPT
SCHEMBL4847288 0.77 IDO1 (0.58) TAAR1IDO1HTR3EHTR3BHTR3A
SCHEMBL793707 0.77 TAAR1 (0.69) PNMTTAAR1DAOGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7462620-B2 Pyrimidinone derivatives and their use in the treatment of atherosclerosis SMITHKLINE BEECHAM, PLC (GB) 2008-12-09 US disclosed
US-20060241126-A1 Pyrimidinone Derivatives and Their Use in the Treatment of Atherosclerosis ELLIOTT RICHARD L 2006-10-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060241126-A1 Pyrimidinone Derivatives and Their Use in the Treatment of Atherosclerosis PLA2G7, PLA2G1B, PLA2G4B PNMT 1157/4885TAAR1 1034/4885DAO 611/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.